A covalent antagonist for the human adenosine A2A receptor

for further investigating covalent interactions at this receptor. It may also serve as a prototype for a therapeutic approach in which a covalent antagonist may be needed to counteract prolonged and persistent presence of the endogenous ligand adenosine. Keywords Gprotein-coupledreceptors .A 2A adenosine receptor .Adenosine .Covalentantagonist ... ................
................