University of Manchester



Novel blood pressure locus and gene discovery using GWAS and expression datasets from blood and the kidneyLouise V. Wain1, Ahmad Vaez2,3, Rick Jansen4, Roby Joehanes5,6, Peter J. van der Most2, A. Mesut Erzurumluoglu1, Paul O'Reilly7, Claudia P. Cabrera8,9, Helen R. Warren8,9, Lynda M. Rose10, Germaine C. Verwoert11, Jouke-Jan Hottenga12, Rona J. Strawbridge13,14, Tonu Esko15,16,17, Dan E. Arking18, Shih-Jen Hwang19,20, Xiuqing Guo21, Zoltan Kutalik22,23, Stella Trompet24,25, Nick Shrine1, Alexander Teumer26,27, Janina S. Ried28, Joshua C. Bis29, Albert V. Smith30,31, Najaf Amin32, Ilja M. Nolte2, Leo-Pekka Lyytik?inen33,34, Anubha Mahajan35, Nicholas J. Wareham36, Edith Hofer37,38, Peter K. Joshi39, Kati Kristiansson40, Michela Traglia41, Aki S. Havulinna40, Anuj Goel42,35, Mike A. Nalls43,44, Siim S?ber45, Dragana Vuckovic46,47, Jian'an Luan36, Fabiola Del Greco M.48, Kristin L. Ayers49, Jaume Marrugat50, Daniela Ruggiero51, Lorna M. Lopez52,53,54, Teemu Niiranen40, Stefan Enroth55, Anne U. Jackson56, Christopher P. Nelson57,58, Jennifer E. Huffman59, Weihua Zhang60,61, Jonathan Marten62, Ilaria Gandin47, Sarah E Harris52,63, Tatijana Zemonik64, Yingchang Lu65, Evangelos Evangelou60,66, Nabi Shah67,68, Martin H. de Borst69, Massimo Mangino70,71, Bram P. Prins72, Archie Campbell73,74, Ruifang Li-Gao75, Ganesh Chauhan76,77, Christopher Oldmeadow78, Gon?alo Abecasis79, Maryam Abedi80, Caterina M. Barbieri41, Michael R. Barnes8,9, Chiara Batini1, John Beilby81,82,83, BIOS Consortium84, Tineka Blake1, Michael Boehnke56, Erwin P. Bottinger65, Peter S. Braund57,58, Morris Brown8,9, Marco Brumat47, Harry Campbell39, John C. Chambers60,61,85, Massimiliano Cocca47, Francis Collins86, John Connell87, Heather J. Cordell88, Jeffrey J. Damman89, Gail Davies52,90, Eco J. de Geus12, Renée de Mutsert75, Joris Deelen91, Yusuf Demirkale92, Alex S.F. Doney67, Marcus D?rr93,27, Martin Farrall42,35, Teresa Ferreira35, Mattias Fr?nberg13,14,94, He Gao60, Vilmantas Giedraitis95, Christian Gieger96, Franco Giulianini10, Alan J. Gow52,97, Anders Hamsten13,14, Tamara B. Harris98, Albert Hofman11,99, Elizabeth G. Holliday78, Jennie Hui81,82,100,83, Marjo-Riitta Jarvelin101,102,103,104, ?sa Johansson55, Andrew D. Johnson6,105, Pekka Jousilahti40, Antti Jula40, Mika K?h?nen106,107, Sekar Kathiresan108,109,110, Kay-Tee Khaw111, Ivana Kolcic112, Seppo Koskinen40, Claudia Langenberg36, Marty Larson6, Lenore J. Launer98, Benjamin Lehne60, David C.M. Liewald52,90, Lifelines Cohort Study113, Li Lin114, Lars Lind115, Fran?ois Mach114, Chrysovalanto Mamasoula116, Cristina Menni70, Borbala Mifsud8, Yuri Milaneschi117, Anna Morgan47, Andrew D. Morris118, Alanna C. Morrison119, Peter J. Munson92, Priyanka Nandakumar18, Quang Tri Nguyen92, Teresa Nutile51, Albertine J. Oldehinkel120, Ben A. Oostra32, Elin Org15, Sandosh Padmanabhan121,74, Aarno Palotie122, Guillaume Paré123, Alison Pattie90, Brenda W.J.H. Penninx117, Neil Poulter124, Peter P. Pramstaller48,125,126, Olli T. Raitakari127,128, Meixia Ren8,129, Kenneth Rice130, Paul M. Ridker10,131, Harri?tte Riese120, Samuli Ripatti122, Antonietta Robino132, Jerome I. Rotter133, Igor Rudan39, Yasaman Saba134, Aude Saint Pierre48,135, Cinzia F. Sala41, Antti-Pekka Sarin122, Reinhold Schmidt37, Rodney Scott78,136,137, Marc A. Seelen69, Denis C. Shields138, David Siscovick139, Rossella Sorice51,140, Alice Stanton141, David J. Stott142, Johan Sundstr?m115, Morris Swertz143, Kent D. Taylor144,145, Simon Thom146, Ioanna Tzoulaki60, Christophe Tzourio76,77,147, André G. Uitterlinden11,148, Understanding Society Scientific group84, Uwe V?ker149,27, Peter Vollenweider150, Sarah Wild39, Gonneke Willemsen12, Alan F. Wright62, Jie Yao21, Sébastien Thériault123, David Conen151, Attia John78,136,137, Peter Sever152, Stéphanie Debette76,77,153, Dennis O. Mook-Kanamori75,154, Eleftheria Zeggini72, Tim D. Spector70, Pim van der Harst155, Colin N.A. Palmer67, Anne-Claire Vergnaud60, Ruth J.F. Loos36,156,157, Ozren Polasek112, John M. Starr52,158, Giorgia Girotto47,46, Caroline Hayward159,74, Jaspal S. Kooner160,61,85, Cecila M. Lindgren17,35, Veronique Vitart59, Nilesh J. Samani57,58, Jaakko Tuomilehto161,162,163,164, Ulf Gyllensten55, Paul Knekt40, Ian J. Deary52,90, Marina Ciullo51,140, Roberto Elosua50, Bernard D. Keavney165, Andrew A. Hicks48, Robert A. Scott36, Paolo Gasparini46,47, Maris Laan45,166, YongMei Liu167, Hugh Watkins42,35, Catharina A. Hartman120, Veikko Salomaa40, Daniela Toniolo41, Markus Perola40,122,168, James F. Wilson39,62, Helena Schmidt134,169, Jing Hua Zhao36, Terho Lehtim?ki33,34, Cornelia M. van Duijn32, Vilmundur Gudnason30,31, Bruce M. Psaty29,170,171,172, Annette Peters28, Rainer Rettig173, Alan James174,175, J Wouter Jukema24, David P. Strachan176, Walter Palmas177, Andres Metspalu15, Erik Ingelsson178,179, Dorret I. Boomsma12, Oscar H. Franco11, Murielle Bochud22, Christopher Newton-Cheh180,108,110,17, Patricia B. Munroe8,9, Paul Elliott104, Daniel I. Chasman10,131, Aravinda Chakravarti18, Joanne Knight181, Andrew P. Morris182,35, Daniel Levy183,20, Martin D. Tobin1, Harold Snieder2*, Mark J. Caulfield8,9*, Georg B. Ehret18,114**: contributing equallyCorresponding authors: Louise V. Wain (louisewain@le.ac.uk) and Georg B. Ehret (georg@rhone.ch)AFFILIATIONS1. Department of Health Sciences, University of Leicester, Leicester LE1 7RH, UK2. Department of Epidemiology, University of Groningen, University Medical Center Groningen, Hanzeplein 1, 9713 GZ Groningen, The Netherlands3. Research Institute for Primordial Prevention of Non-communicable Disease, Isfahan University of Medical Sciences, Isfahan, Iran4. Department of Psychiatry, VU University Medical Center, Neuroscience Campus Amsterdam, Amsterdam, The Netherlands5. Hebrew SeniorLife, Harvard Medical School, 1200 Centre Street Room #609, Boston, MA 02131, USA6. National Heart, Lung and Blood Institute's Framingham Heart Study, Framingham, MA 01702, USA7. Institute of Psychiatry, Psychology and Neuroscience, King's College London, London SE5 8AF, UK8. Clinical Pharmacology, William Harvey Research Institute, Barts and The London School of Medicine and Dentistry, Queen Mary University of London, London, EC1M 6BQ, UK9. NIHR Barts Cardiovascular Biomedical Research Unit, Barts and The London School of Medicine and Dentistry, Queen Mary University of London, London, EC1M 6BQ, UK10. Division of Preventive Medicine, Brigham and Women's Hospital, Boston MA 02215, USA11. Department of Epidemiology, Erasmus MC, Rotterdam, 3000CA, The Netherlands12. Department of Biological Psychology, Vrije Universiteit, Amsterdam, EMGO+ institute, VU University medical center, Amsterdam, The Netherlands13. Cardiovascular Medicine Unit, Department of Medicine Solna, Karolinska Institutet, Stockholm, 17176, Sweden14. Centre for Molecular Medicine, Karolinska Universitetsjukhuset, Solna, 171 76, Sweden15. Estonian Genome Center, University of Tartu, Tartu, 51010, Estonia16. Divisions of Endocrinology/Children's Hospital, Boston, MA 02115, USA17. Broad Institute of Harvard and MIT, Cambridge, MA 02139 USA18. Center for Complex Disease Genomics, McKusick-Nathans Institute of Genetic Medicine, Johns Hopkins University School of Medicine, Baltimore, MD 21205, USA19. The Population Science Branch, Division of Intramural Research, National Heart Lung and Blood Institute national Institute of Health, Bethesda, MD 20892, USA20. The Framingham Heart Study, Framingham MA 01702, USA21. The Institute for Translational Genomics and Population Sciences, Department of Pediatrics, LABioMed at Harbor-UCLA Medical Center, 1124 W. Carson Street, Torrance, CA 90502, USA22. Institute of Social and Preventive Medicine, Lausanne University Hospital, Route de la Corniche 10, 1010 Lausanne, Switzerland23. Swiss Institute of Bioinformatics, Lausanne, Switzerland24. Department of Cardiology, Leiden University Medical Center, Leiden, 2300RC, The Netherlands25. Department of Gerontology and Geriatrics, Leiden University Medical Center, Leiden, 2300RC, The Netherlands26. Institute for Community Medicine, University Medicine Greifswald, Greifswald, 17475, Germany27. DZHK (German Centre for Cardiovascular Research), partner site Greifswald, Greifswald, 17475, Germany28. Institute of Epidemiology II, Helmholtz Zentrum München, Neuherberg 85764, Germany29. Cardiovascular Health Research Unit, Department of Medicine, University of Washington, Seattle, WA 98101, USA30. Icelandic Heart Assoication, Kopavogur, Iceland31. Faculty of Medicine, University of Iceland, Reykjavik, Iceland32. Genetic Epidemiology Unit, Department of Epidemiology, Erasmus MC, Rotterdam, 3000CA, The Netherlands33. Department of Clinical Chemistry, Fimlab Laboratories, Tampere 33520, Finland34. Department of Clinical Chemistry, Faculty of Medicine and Life Sciences, University of Tampere, Tampere 33014, Finland35. Wellcome Trust Centre for Human Genetics, University of Oxford, Roosevelt Drive, Oxford OX3 7BN, UK36. MRC Epidemiology Unit, University of Cambridge School of Clinical Medicine, Institute of Metabolic Science, Cambridge Biomedical Campus, Cambridge, CB2 0QQ, UK37. Clinical Division of Neurogeriatrics, Department of Neurology, Medical University Graz, Auenbruggerplatz 22, 8036 Graz, Austria38. Institute of Medical Informatics, Statistics and Documentation, Medical University Graz, Auenbruggerplatz 2, 8036 Graz, Austria39. Centre for Global Health Research, Usher Institute of Population Health Sciences and Informatics, University of Edinburgh EH89AG, Scotland, UK40. Department of Health, National Institute for Health and Welfare (THL), Helsinki, Finland41. Division of Genetics and Cell Biology, San Raffaele Scientific Institute, 20132 Milano, Italy42. Division of Cardiovascular Medicine, Radcliffe Department of Medicine, University of Oxford, Oxford, OX3 9DU, UK43. Laboratory of Neurogenetics, National Institute on Aging, NIH, Bethesda, 20892, USA44. Kelly Services, Rockville, MD, USA45. Human Molecular Genetics Research Group, Institute of Molecular and Cell Biology, University of Tartu, Riia St.23, 51010 Tartu, Estonia46. Experimental Genetics Division, Sidra Medical and Research Center, PO Box 26999, Doha, Qatar47. Department of Medical, Surgical and Health Sciences, University of Trieste, Strada di Fiume 447, Trieste, 34100, Italy48. Center for Biomedicine, European Academy Bozen/Bolzano (EURAC), Bolzano, Italy - Affiliated Institute of the University of Lübeck, Germany49. Department of Genetics and Genomic Sciences, Icahn School of Medicine at Mount Sinai, New York, NY, USA50. Cardiovascular Epidemiology and Genetics, IMIM. Dr Aiguader 88, Barcelona, 08003, Spain51. Institute of Genetics and Biophysics A. Buzzati-Traverso, CNR, via P. Castellino 111, 80131 Napoli, Italy52. Centre for Cognitive Ageing and Cognitive Epidemiology, University of Edinburgh, 7 George Square, Edinburgh EH8 9JZ, UK53. Department of Psychiatry, Royal College of Surgeons in Ireland, Education and Research Centre, Beaumont Hospital, Dublin, Ireland54. University College Dublin, UCD Conway Institute, Centre for Proteome Research, UCD, Belfield, Dublin, Ireland55. Department of Immunology, Genetics and Pathology, Uppsala Universitet, Science for Life Laboratory, Husargatan 3, Uppsala, SE-75108, Sweden56. Department of Biostatistics and Center for Statistical Genetics, University of Michigan, Ann Arbor, MI 48109, USA57. Department of Cardiovascular Sciences, University of Leicester, Leicester LE3 9QP, UK58. NIHR Leicester Cardiovascular Biomedical Research Unit, Glenfield Hospital, Leicester LE3 9QP, UK59. MRC Human Genetics Unit, IGMM, University of Edinburgh, Western General Hospital, Edinburgh, EH4 2XU Scotland, UK60. Department of Epidemiology and Biostatistics, School of Public Health, Imperial College London, London W2 1PG, United Kingdom61. Department of Cardiology, Ealing Hospital NHS Trust, Uxbridge Road, Southall, Middlesex UB1 3EU, UK62. MRC Human Genetics Unit, Institute of Genetics and Molecular Medicine, University of Edinburgh, Western General Hospital, Crewe Road, Edinburgh, EH4 2XU, UK63. Medical Genetics Section, University of Edinburgh Centre for Genomic and Experimental Medicine and MRC Institute of Genetics and Molecular Medicine, Western General Hospital, Crewe Road, Edinburgh EH4 2XU, UK64. Department of Biology, Faculty of Medicine, University of Split, Croatia65. The Charles Bronfman Institute for Personalized Medicine, Icachn School of Medicine at Mount Sinai, New York, NY 10029, USA66. Department of Hygiene and Epidemiology, University of Ioannina Medical School, Ioannina, 45110, Greece67. Medical Research Institute, University of Dundee, Ninewells Hospital and Medical School, Dundee, DD1 9SY, Scotland, UK68. Department of Pharmacy, COMSATS Institute of Information Technology, Abbottabad, 22060, Pakistan69. Department of Internal Medicine, Division of Nephrology, University of Groningen, University Medical Center Groningen, PO Box 30001, 9700 RB Groningen, The Netherlands70. Department of Twin Research and Genetic Epidemiology, King’s College London, Lambeth Palace Rd, London, SE1 7EH, UK71. National Institute for Health Research Biomedical Research Centre, London SE1 9RT, UK72. Department of Human Genetics, Wellcome Trust Sanger Institute, CB10 1HH, United Kingdom73. Medical Genetics Section, Centre for Genomic and Experimental Medicine, Institute of Genetics and Molecular Medicine, University of Edinburgh, Edinburgh EH4 2XU, UK74. Generation Scotland, Centre for Genomic and Experimental Medicine, University of Edinburgh, Edinburgh, EH4 2XU, UK75. Department of Clinical Epidemiology, Leiden University Medical Center, Leiden, The Netherlands76. INSERM U 1219, Bordeaux Population Health center, Bordeaux, France77. Bordeaux University, Bordeaux, France78. Hunter Medical Research Institute, New Lambton, NSW 2305, Australia79. Center for Statistical Genetics, Dept. of Biostatistics, SPH II, 1420 Washington Heights, Ann Arbor, MI 48109-2029, USA80. Department of Genetics and Molecular Biology, Isfahan University of Medical Sciences, Isfahan, Iran81. Busselton Population Medical Research Institute, Western Australia82. PathWest Laboratory Medicine of Western Australia, NEDLANDS, Western Australia83. School of Pathology and Laboratory Medicine, The University of Western Australia, NEDLANDS, Western Australia84. For a complete list of contributing authors, please see Supporting Information.85. Imperial College Healthcare NHS Trust, London, UK86. Medical Genomics and Metabolic Genetics Branch, National Human Genome Research Institute, NIH, Bethesda, MD 20892, USA87. University of Dundee, Ninewells Hospital & Medical School, Dundee, DD1 9SY, UK88. Institute of Genetic Medicine, Newcastle University, Newcastle upon Tyne, UK89. Department of Pathology, Amsterdam Medical Center, Meibergdreef 9, 1105 AZ, Amsterdam, The Netherlands90. Department of Psychology, University of Edinburgh, 7 George Square, Edinburgh, EH8 9JZ, UK91. Department of Molecular Epidemiology, Leiden University Medical Center, Leiden, 2300RC, The Netherlands92. Center for Information Technology, NIH, USA93. Department of Internal Medicine B, University Medicine Greifswald, Greifswald, 17475, Germany94. Department of Numerical Analysis and Computer Science, Stockholm University, Lindstedtsv?gen 3, Stockholm, 100 44, Sweden95. Department of Public Health and Caring Sciences, Geriatrics, Uppsala 752 37, Sweden96. Helmholtz Zentrum Muenchen, Deutsches Forschungszentrum fuer Gesundheit und Umwelt (GmbH), Ingolstaedter Landstr. 1, 85764 Neuherberg, München, Germany97. Department of Psychology, School of Life Sciences, Heriot-Watt University, Edinburgh, EH14 4AS, UK98. Intramural Research Program, Laboratory of Epidemiology, Demography, and Biometry, National Institute on Aging, USA99. Department of Epidemiology, Harvard T.H. Chan School of Public Health, Boston, MA 02115, USA100. School of Population and Global Health, The University of Western Australia, NEDLANDS, Western Australia101. Center For Life-course Health Research, P.O. Box 5000, FI-90014 University of Oulu, Finland102. Biocenter Oulu, P.O. Box 5000, Aapistie 5A, FI-90014 University of Oulu, Finland103. Unit of Primary Care, Oulu University Hospital, Kajaanintie 50, P.O. Box 20, FI-90220 Oulu, 90029 OYS, Finland104. MRC-PHE Centre for Environment and Health, Department of Epidemiology and Biostatistics, School of Public Health, Imperial College London, Norfolk Place, W2 1PG London, UK105. National Heart, Lung and Blood Institute, Cardiovascular Epidemiology and Human Genomics Branch, Bethesda, MD 20814, USA106. Department of Clinical Physiology, Tampere University Hospital, Tampere 33521, Finland107. Department of Clinical Physiology, Faculty of Medicine and Life Sciences, University of Tampere, Tampere 33014, Finland108. Cardiovascular Research Center, Massachusetts General Hospital, Boston, MA 02114, USA109. Center for Human Genetics, Massachusetts General Hospital, 185 Cambridge Street, Boston, MA 02114, USA110. Program in Medical and Population Genetics, Broad Institute, 7 Cambridge Center, Cambridge, MA 02142, USA111. Department of Public Health and Primary Care, Institute of Public Health, University of Cambridge, Cambridge CB2 2SR, UK112. Department of Public Health, Faculty of Medicine, University of Split, Croatia113. See complete listing of contributors in the Supporting Information.114. Cardiology, Department of Medicine, Geneva University Hospital, Rue Gabrielle-Perret-Gentil 4, 1211 Geneva 14, Switzerland115. Department of Medical Sciences, Cardiovascular Epidemiology, Uppsala University, Uppsala 751 85, Sweden116. Institute of Health and Society, Newcastle University, Newcastle upon Tyne, UK117. Department of Psychiatry, EMGO Institute for Health and Care Research, VU University Medical Center, A.J. Ernststraat 1187, 1081 HL Amsterdam, The Netherlands118. School of Molecular, Genetic and Population Health Sciences, University of Edinburgh, Medical School,Teviot Place, Edinburgh, EH8 9AG, Scotland, UK119. Department of Epidemiology, Human Genetics and Environmental Sciences, School of Public Health, University of Texas Health Science Center at Houston, 1200 Pressler St., Suite 453E, Houston, TX 77030, USA120. Interdisciplinary Center Psychopathology and Emotion Regulation (IPCE), University of Groningen, University Medical Center Groningen, Hanzeplein 1, PO Box 30001, 9700 RB Groningen, The Netherlands121. British Heart Foundation Glasgow Cardiovascular Research Centre, Institute of Cardiovascular and Medical Sciences, College of Medical, Veterinary and Life Sciences, University of Glasgow, Glasgow G12 8TA, UK122. Institute for Molecular Medicine Finland (FIMM), University of Helsinki, Helsinki, Finland123. Department of Pathology and Molecular Medicine, McMaster University, 1280 Main St W, Hamilton, L8S 4L8, Canada124. School of Public Health, Imperial College London, W2 1PG, UK125. Department of Neurology, General Central Hospital, Bolzano, Italy126. Department of Neurology, University of Lübeck, Lübeck, Germany127. Department of Clinical Physiology and Nuclear Medicine, Turku University Hospital, Turku 20521, Finland128. Research Centre of Applied and Preventive Cardiovascular Medicine, University of Turku, Turku 20014, Finland129. Department of?Cardiology,?Fujian Provincial Hospital, Fujian Medical University, Fuzhou 350001, China130. Department of Biostatistics University of Washington, Seattle, WA 98101, USA131. Harvard Medical School, Boston MA, USA132. Institute for Maternal and Child Health IRCCS Burlo Garofolo, Via dell'Istria 65, Trieste, 34200, Italy133. The Institute for Translational Genomics and Population Sciences, Departments of Pediatrics and Medicine, LABioMed at Harbor-UCLA Medical Center, 1124 W. Carson Street, Torrance, CA 90502, USA134. Institute of Molecular Biology and Biochemistry, Centre for Molecular Medicine, Medical University of Graz, Harrachgasse 21, 8010 Graz, Austria135. INSERM U1078, Etablissement Fran?ais du Sang, 46 rue Félix Le Dantec, CS 51819, Brest Cedex 2 29218, France136. Faculty of Health, University of Newcastle, Callaghan NSW 2308, Australia137. John Hunter Hospital, New Lambton NSW 2305, Australia138. School of Medicine, Conway Institute, University College Dublin, Ireland139. The New York Academy of Medicine. 1216 5th Ave, New York, NY 10029, USA140. IRCCS Neuromed, Pozzilli, Isernia, Italy141. Molecular and Cellular Therapeutics, Royal College of Surgeons in Ireland, Dublin 2, Ireland142. Institute of Cardiovascular and Medical Sciences, Faculty of Medicine, University of Glasgow, United Kingdom143. Department of Genetics, University of Groningen, University Medical Center Groningen, PO Box 30001, 9700 RB Groningen, The Netherlands144. Institute for Translational Genomics and Population Sciences. Los Angeles BioMedical Research Institute at Harbor-UCLA Medical Center, Torrance, CA, 90502, USA145. Division of Genetic Outcomes, Department of Pediatrics, Harbor-UCLA Medical Center, Torrance, CA, 90502, USA146. International Centre for Circulatory Health, Imperial College London, W2 1PG, UK147. Department of Public Health, Bordeaux University Hospital, Bordeaux, France148. Department of Internal Medicine, Erasmus MC, Rotterdam, 3000CA, The Netherlands149. Interfaculty Institute for Genetics and Functional Genomics, University Medicine Greifswald, Greifswald, 17475, Germany150. Department of Internal Medicine, Lausanne Universiyt Hospital, CHUV, 1011 Lausanne, Switzerland151. Population Health Research Institute, McMaster University, Hamilton Ontario, Canada152. National Heart and Lung Institute, Imperial College London, W2 1PG, UK153. Department of Neurology, Bordeaux University Hospital, Bordeaux, France154. Department of Public Health and Primary Care, Leiden University Medical Center, Leiden, The Netherlands155. Department of Cardiology, University of Groningen, University Medical Center Groningen, PO Box 30001, 9700 RB Groningen, The Netherlands156. The Charles Bronfman Institute for Personalized Medicine, The Icahn School of Medicine at Mount Sinai, New York, NY 10029, USA157. Mindich Child health Development Institute, The Icahn School of Medicine at Mount Sinai, New York, NY 10029, USA158. Alzheimer Scotland Dementia Research Centre, University of Edinburgh, 7 George Square, Edinburgh, EH8 9JZ, UK159. Medical Research Council Human Genetics Unit, Institute of Genetics and Molecular Medicine, University of Edinburgh, Edinburgh EH4 2XU, UK160. National Heart and Lung Institute, Imperial College London, Hammersmith Hospital Campus, Du Cane Road, London W12 0NN, UK161. Diabetes Prevention Unit, National Institute for Health and Welfare, 00271 Helsinki, Finland162. South Ostrobothnia Central Hospital, 60220 Sein?joki, Finland163. Red RECAVA Grupo RD06/0014/0015, Hospital Universitario La Paz, 28046 Madrid, Spain164. Centre for Vascular Prevention, Danube-University Krems, 3500 Krems, Austria165. Institute of Cardiovascular Sciences, The University of Manchester, Manchester, UK166. Institute of Biomedicine and Translational Medicine, University of Tartu, Ravila Str. 19, 50412 Tartu, Estonia167. Division of Public?Health?Sciences, Wake Forest School of Medicine, Winston-Salem, 27106, USA168. University of Tartu, Tartu, Estonia169. Department of Neurology, Medical University Graz, Auenbruggerplatz 22, 8036 Graz, Austria170. Department of Epidemiology University of Washington, Seattle, WA 98101, USA171. Department of Health Services, University of Washington, Seattle, WA 98101, USA172. Group Health Research Institute, Group Health, Seattle, WA, 98101, USA173. Institute of Physiology, University Medicine Greifswald, Karlsburg, 17495, Germany174. Department of Pulmonary Physiology and Sleep, Sir Charles Gairdner Hospital, Hospital Avenue, Nedlands 6009,H57, Western Australia175. School of Medicine and Pharmacology, University of Western Australia, Australia176. Population Health Research Institute, St George's, University of London, London SW17 0RE, UK177. Department of Medicine, Columbia University Medical Center, 622 West 168th Street, PH 9, East, 107, New York, NY 10032, USA178. Department of Medical Sciences, Molecular Epidemiology and Science for Life Laboratory, Uppsala University, Uppsala 752 37, Sweden179. Department of Medicine, Division of Cardiovascular Medicine, Stanford University School of Medicine, Stanford, CA 94305, USA180. Center for Human Genetic Research, Massachusetts General Hospital, Boston, MA 02114, USA181. Data Science Institute and Lancaster Medical School, Lancaster University, LA1 4YG, UK182. Department of Biostatistics, University of Liverpool, Block F, Waterhouse Building, 1-5 Brownlow Street, Liverpool L69 3GL, UK183. The population Science Branch, Division of Intramural Research, National Heart Lung and Blood Institute national Institute of Health, Bethesda MD 20892, USACorresponding authors: Louise V. Wain (louisewain@le.ac.uk) and Georg B. Ehret (georg@jhmi.edu)ABSTRACTElevated blood pressure is a major risk factor for cardiovascular disease and has a substantial genetic contribution. Genetic variation influencing blood pressure has the potential to identify new pharmacological targets for the treatment of hypertension. To discover additional novel blood pressure loci, we used 1000 Genomes Project-based imputation in 150,134 European ancestry individuals and sought significant evidence for independent replication in a further 228,245 individuals. We report 6 new signals of association in or near HSPB7, TNXB, LRP12, LOC283335, SEPT9 and AKT2, and provide new replication evidence for a further 2 signals in EBF2 and NFKBIA. Combining large whole-blood gene expression resources totaling 12,607 individuals, we investigated all novel and previously reported signals and identified 48 genes with evidence for involvement in BP regulation that are significant in multiple resources. Three novel kidney-specific signals were also detected. These robustly implicated genes may provide new leads for therapeutic innovation.INTRODUCTIONGenetic support for a drug target increases the likelihood of success in drug development PEVuZE5vdGU+PENpdGU+PEF1dGhvcj5OZWxzb248L0F1dGhvcj48WWVhcj4yMDE1PC9ZZWFyPjxS

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ZT5=

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ADDIN EN.CITE.DATA 2. A number of large studies have described blood pressure (BP) variant identification by genome-wide and targeted association approaches eEQ7RGVwYXJ0bWVudCBvZiBDYXJkaW9sb2d5LCBMZWlkZW4gVW5pdmVyc2l0eSBNZWRpY2FsIENl

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ADDIN EN.CITE.DATA 3-19. Clinically the most predictive BP traits for cardiovascular risk are systolic blood pressure (SBP) and diastolic blood pressure (DBP), reflecting roughly the peak and trough of the BP curve, and pulse pressure (PP), the difference between SBP and DBP ADDIN EN.CITE <EndNote><Cite><Author>Safar</Author><Year>2012</Year><RecNum>17</RecNum><DisplayText><style face="superscript">20</style></DisplayText><record><rec-number>17</rec-number><foreign-keys><key app="EN" db-id="2fxv5r22r55ep6e05xs5xxv2rae52rztt2vr" timestamp="1473414867">17</key></foreign-keys><ref-type name="Journal Article">17</ref-type><contributors><authors><author>Safar, M. E.</author><author>Nilsson, P. M.</author><author>Blacher, J.</author><author>Mimran, A.</author></authors></contributors><auth-address>Paris Descartes University; AP-HP; Diagnosis and Therapeutic Center, Hotel-Dieu, 1, place du Parvis Notre-Dame, 75181, Paris Cedex 04, France. michel.safar@htd.aphp.fr</auth-address><titles><title>Pulse pressure, arterial stiffness, and end-organ damage</title><secondary-title>Curr Hypertens Rep</secondary-title></titles><periodical><full-title>Curr Hypertens Rep</full-title></periodical><pages>339-44</pages><volume>14</volume><number>4</number><keywords><keyword>Arteries/*pathology</keyword><keyword>Blood Pressure/*physiology</keyword><keyword>Endothelium, Vascular/*pathology</keyword><keyword>Humans</keyword><keyword>Hypertension/*complications/pathology</keyword><keyword>Renal Insufficiency/etiology/pathology</keyword><keyword>Risk</keyword><keyword>Stress, Physiological</keyword><keyword>Vascular Resistance/*physiology</keyword><keyword>Vascular Stiffness/*physiology</keyword></keywords><dates><year>2012</year><pub-dates><date>Aug</date></pub-dates></dates><isbn>1534-3111 (Electronic)&#xD;1522-6417 (Linking)</isbn><accession-num>22555981</accession-num><urls><related-urls><url> reflecting arterial stiffness. Using these three traits, we undertook a meta-analysis of 150,134 individuals from 54 genome-wide association studies of European ancestry with imputation based on the 1000 Genomes Project Phase 1. To minimize reporting of false positive associations, we sought stringent evidence for significant independent replication in a further 228,245 individuals. We further followed up novel and previously reported association signals in multiple large gene expression databases and the largest kidney tissue gene expression resource currently available. Finally, we searched for enrichment of associated genes in biological pathways and gene sets and identified whether any of the genes were known drug targets or had tool molecules.MATERIALS AND METHODSStudies Stage 1Results from 54 independent European-ancestry studies, totaling 150,134 individuals, were included in the Stage 1 meta-analysis: AGES (n=3215), ARIC (n=9402), ASPS (n=828), B58C (n=6458), BHS (n=4492), CHS (n=3254), Cilento study (n=999), COLAUS (n=5404), COROGENE-CTRL (n=1878), CROATIA-Vis (n=945), CROATIA-Split (n=494), CROATIA-Korcula (n=867), EGCUT (n=6395), EGCUT2 (n=1844), EPIC (n=2100), ERF (n=2617), Fenland (n=1357), FHS (n=8096), FINRISK-ctrl (n=861), FINRISK CASE (n=839), FUSION (n=1045), GRAPHIC (n=1010), H2000-CTRL (n=1078), HealthABC (n=1661), HTO (n=1000), INGI-CARL (n=456), INGI-FVG (n=746), INGI-VB (n=1775), IPM (n=300), KORAS3 (n=1590), KORAS4 (n=3748), LBC1921 (n=376), LBC1936 (n=800), LOLIPOP-EW610 (n=927), MESA (n=2678), MICROS (n=1148), MIGEN (n=1214), NESDA (n=2336), NSPHS (n=1005), NTR (n=1490), PHASE (n=4535), PIVUS (n=945), PROCARDIS (n=1652), SHIP (n=4068), ULSAM (n=1114), WGHS (n=23049), YFS (n=1987), ORCADES (n=1908), RS1 (n=5645), RS2 (n=2152), RS3 (n=3018), TRAILS (n=1262), TRAILS-CC (n=282) and TWINGENE (n=9789). Full study names and general study information is given in Supplementary Table 1.Study-level genotyping and association testingThree quantitative BP traits were analyzed: SBP, DBP, and PP (difference between SBP and DBP). Within each study, individuals known to be taking anti-hypertensive medication had 15 mmHg added to their raw SBP value and 10 mmHg added to their raw DBP values ADDIN EN.CITE <EndNote><Cite><Author>Tobin</Author><Year>2005</Year><RecNum>37</RecNum><DisplayText><style face="superscript">21</style></DisplayText><record><rec-number>37</rec-number><foreign-keys><key app="EN" db-id="2fxv5r22r55ep6e05xs5xxv2rae52rztt2vr" timestamp="1474688750">37</key></foreign-keys><ref-type name="Journal Article">17</ref-type><contributors><authors><author>Tobin, M. D.</author><author>Sheehan, N. A.</author><author>Scurrah, K. J.</author><author>Burton, P. R.</author></authors></contributors><auth-address>Biostatistics and Genetic Epidemiology, Department of Health Sciences, University of Leicester, 22-28 Princess Road West, Leicester LE1 6TP, U.K. mt47@leicester.ac.uk</auth-address><titles><title>Adjusting for treatment effects in studies of quantitative traits: antihypertensive therapy and systolic blood pressure</title><secondary-title>Stat Med</secondary-title></titles><periodical><full-title>Stat Med</full-title></periodical><pages>2911-35</pages><volume>24</volume><number>19</number><keywords><keyword>Aged</keyword><keyword>Antihypertensive Agents/*pharmacology</keyword><keyword>Bias (Epidemiology)</keyword><keyword>Blood Pressure/drug effects/*genetics</keyword><keyword>Computer Simulation</keyword><keyword>Female</keyword><keyword>Humans</keyword><keyword>Male</keyword><keyword>Middle Aged</keyword><keyword>*Models, Genetic</keyword><keyword>*Models, Statistical</keyword><keyword>*Quantitative Trait, Heritable</keyword></keywords><dates><year>2005</year><pub-dates><date>Oct 15</date></pub-dates></dates><isbn>0277-6715 (Print)&#xD;0277-6715 (Linking)</isbn><accession-num>16152135</accession-num><urls><related-urls><url>. A summary of BP phenotypes in each study is given in Supplementary Table 2. Association testing was undertaken according to a central analysis plan that specified the use of sex, age, age2, and body mass index (BMI) as covariates and optional inclusion of additional covariates to account for population stratification (Supplementary Table 3). Trait residuals were calculated for each trait using a normal linear regression of the medication-adjusted trait values (mmHg) onto all covariates. The genotyping array, pre-imputation quality control filters, imputation software and association testing software used by each study are listed in Supplementary Table 4. All studies imputed to the 1000 Genomes Project Phase 1 integrated release version 3 [March 2012] all ancestry reference panel PEVuZE5vdGU+PENpdGU+PEF1dGhvcj5HZW5vbWVzIFByb2plY3Q8L0F1dGhvcj48WWVhcj4yMDEy

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ADDIN EN.CITE.DATA 22. Imputed genotype dosages were used to take into account uncertainty in the imputation. Association testing was carried out using linear regression of the trait residuals onto genotype dosages under an additive genetic model. Methods to account for relatedness within a study were used where appropriate (Supplementary Table 3). Results for all variants (SNPs and INDELs) were then returned to the central analysis group for further quality control checks and meta-analysis.Stage 1 meta-analysisCentral quality control checks were undertaken across all results sets. This included checks to ensure allele frequency consistency (across studies and with reference populations), checks of effect size and standard error distributions (i.e. to highlight phenotype issues) and generation of quantile-quantile (QQ) plots and genomic inflation factor lambdas to check for over- or under-inflation of test statistics. Genomic control was applied (if lambda>1) at study-level. Variants with imputation quality <0.3 were excluded prior to meta-analysis. Inverse variance weighted meta-analysis was undertaken. After meta-analysis, variants with a weighted minor allele frequency of less than 1 % or N effective (product of study sample size and imputation quality summed across contributing studies) <60% were then excluded and meta-analysis genomic control lambda calculated and used to adjust the meta-analysis results. Selection of regions for follow-upFor each trait, regions of association were selected by ranking variants by P value, recording the variant with the lowest P value as a sentinel variant and then excluding all variants +/-500kb from the sentinel and re-ranking the remaining variants. This was undertaken iteratively until all sentinel variants representing 1Mb regions containing associations with P <10-6 had been identified. To identify additional signals represented by secondary sentinel variants within 500kb of each of the sentinel variants, GCTA ADDIN EN.CITE <EndNote><Cite><Author>Yang</Author><Year>2011</Year><RecNum>77</RecNum><DisplayText><style face="superscript">23</style></DisplayText><record><rec-number>77</rec-number><foreign-keys><key app="EN" db-id="2fxv5r22r55ep6e05xs5xxv2rae52rztt2vr" timestamp="1475220087">77</key></foreign-keys><ref-type name="Journal Article">17</ref-type><contributors><authors><author>Yang, J.</author><author>Lee, S. H.</author><author>Goddard, M. E.</author><author>Visscher, P. M.</author></authors></contributors><auth-address>Queensland Statistical Genetics Laboratory, Queensland Institute of Medical Research, 300 Herston Road, Brisbane, Queensland 4006, Australia. jian.yang@qimr.edu.au</auth-address><titles><title>GCTA: a tool for genome-wide complex trait analysis</title><secondary-title>Am J Hum Genet</secondary-title></titles><periodical><full-title>Am J Hum Genet</full-title><abbr-1>American journal of human genetics</abbr-1></periodical><pages>76-82</pages><volume>88</volume><number>1</number><keywords><keyword>Chromosomes, Human, X/*genetics</keyword><keyword>Computer Simulation</keyword><keyword>Dosage Compensation, Genetic</keyword><keyword>Female</keyword><keyword>Genetic Linkage</keyword><keyword>Genome-Wide Association Study/*methods</keyword><keyword>Humans</keyword><keyword>Male</keyword><keyword>Models, Genetic</keyword><keyword>*Polymorphism, Single Nucleotide</keyword><keyword>*Quantitative Trait Loci</keyword><keyword>*Software</keyword></keywords><dates><year>2011</year><pub-dates><date>Jan 7</date></pub-dates></dates><isbn>1537-6605 (Electronic)&#xD;0002-9297 (Linking)</isbn><accession-num>21167468</accession-num><urls><related-urls><url> was used to run conditional analyses (conditioned on the first sentinel variant) on each of the 1Mb regions using GWAS summary statistics and LD information from ARIC. This was done both for putatively novel regions and for regions that had previously been reported. A chi-squared test of heterogeneity of effect sizes across the 54 studies was run for each sentinel variant and those with P <0.05 for heterogeneity were excluded from further follow-up. Variants with P <10-6 after conditioning on the sentinel SNP (novel or known) in the region and for which any attenuation of the –log10 P value was less than 1.5 fold, were also taken forward for replication.Studies stage 2Data from 14 independent studies, totaling 87,360 individuals, and the first release of UK Biobank, totaling 140,886 individuals, were combined to replicate the findings from stage 1 (i.e. totaling 228,245 individuals). Stage 2 study details, including full study names, are given in Supplementary Table 6 and included 3C-Dijon (n=4061), Airwave (n=14023), ASCOT-SC (n=2462), ASCOT-UK (n=3803), BRIGHT (n=1791), GAPP (n=1685), GoDARTs (n=7413), GS:SFHS (n=9749), HCS (n=2112), JUPITER (n=8718), LifeLines (n=13376), NEO (n=5731), TwinsUK (n=4973), UK Biobank-CMC (n=140,886) and UKHLS (n=7462). Analysis was undertaken using the same methods as described for Stage 1 studies. UK Biobank-CMC utilized a newer imputation reference panel than the other studies and where a requested variant was not available, a proxy was used (next most significant P value with linkage disequilibrium r2> 0.6 with original top variant). Results from all stage 2 studies were meta-analyzed using inverse-variance weighted meta-analysis. Two of the variants, rs1048238 and chr1:243458005:I, were not available in the largest study in Stage 2 (UK Biobank-CMC) and so proxy variants were selected (based on P value and LD).Stage 1 + Stage 2 meta-analysisFollowing meta-analysis of stage 1 and stage 2 results, signals with a P > 5x10-8 were excluded. Of the signals with a final P <5x10-8, support for independent replication within the stage 2 studies only was sought. Any signals which had P < 5x10-8 and evidence for independent replication in stage 2 alone, indicated by P < 8.2x10-4 (Bonferroni correction for 61 tests) were reported as novel signals of association with BP. Any signals which were subsequently reported by other BP GWAS that were accepted for publication during the time this analysis was ongoing, or signals for which independence from another known signal could not be established, were removed from our list of novel signals at this stage (Supplementary Table 5).Genotype and gene expressionWe searched for signals of association of genotype with gene expression for the 22 signals (including 8 novel) signals described in this study (Supplementary Table 7) and all signals reported prior to our study (Supplementary Table 10) dGVyIE91bHUsIFVuaXZlcnNpdHkgb2YgT3VsdSwgT3VsdSwgRmlubGFuZC4mI3hEO0NlbnRlciBm

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ADDIN EN.CITE.DATA 3-17, 24 in 3 whole-blood data sets, 1 kidney data set and the GTEx multiple tissue data resource, which included whole-blood ADDIN EN.CITE <EndNote><Cite><Author>Consortium</Author><Year>2015</Year><RecNum>28</RecNum><DisplayText><style face="superscript">25</style></DisplayText><record><rec-number>28</rec-number><foreign-keys><key app="EN" db-id="2fxv5r22r55ep6e05xs5xxv2rae52rztt2vr" timestamp="1474022265">28</key></foreign-keys><ref-type name="Journal Article">17</ref-type><contributors><authors><author>G. TEx Consortium</author></authors></contributors><titles><title>Human genomics. The Genotype-Tissue Expression (GTEx) pilot analysis: multitissue gene regulation in humans</title><secondary-title>Science</secondary-title></titles><periodical><full-title>Science</full-title></periodical><pages>648-60</pages><volume>348</volume><number>6235</number><keywords><keyword>Alleles</keyword><keyword>Blood Pressure/genetics</keyword><keyword>Disease/*genetics</keyword><keyword>GTPase-Activating Proteins/genetics</keyword><keyword>*Gene Expression Regulation</keyword><keyword>Gene Regulatory Networks</keyword><keyword>*Genetic Variation</keyword><keyword>Genome, Human/*genetics</keyword><keyword>Genome-Wide Association Study</keyword><keyword>Genotype</keyword><keyword>Humans</keyword><keyword>Multigene Family</keyword><keyword>Organ Specificity/genetics</keyword><keyword>Pilot Projects</keyword><keyword>*Quantitative Trait Loci</keyword><keyword>RNA Splicing</keyword><keyword>RNA, Untranslated/genetics</keyword><keyword>Sequence Analysis, RNA</keyword><keyword>Tibial Arteries/metabolism</keyword><keyword>*Transcriptome</keyword></keywords><dates><year>2015</year><pub-dates><date>May 8</date></pub-dates></dates><isbn>1095-9203 (Electronic)&#xD;0036-8075 (Linking)</isbn><accession-num>25954001</accession-num><urls><related-urls><url>. We selected cis signals of association which were significant after controlling for 5% False Discovery Rate (FDR). The 3 whole-blood eQTL data sets were the NHLBI Systems Approach to Biomarker Research in Cardiovascular Disease initiative whole-blood eQTL resource (SABRe) (microarray, n=5257), NESDA-NTR (microarray, n=4896), BIOS (RNAseq, n=2116). The whole-blood data from GTEx was based on data from 338 samples. The kidney data set comprised 236 donor-kidney samples from 134 donors PEVuZE5vdGU+PENpdGU+PEF1dGhvcj5EYW1tYW48L0F1dGhvcj48WWVhcj4yMDE1PC9ZZWFyPjxS

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ADDIN EN.CITE.DATA 26. Full details of each data set can be found in the Supporting Information. The source transcriptomic renal data as describedPEVuZE5vdGU+PENpdGU+PEF1dGhvcj5EYW1tYW48L0F1dGhvcj48WWVhcj4yMDE1PC9ZZWFyPjxS

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ADDIN EN.CITE PEVuZE5vdGU+PENpdGU+PEF1dGhvcj5EYW1tYW48L0F1dGhvcj48WWVhcj4yMDE1PC9ZZWFyPjxS

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ADDIN EN.CITE.DATA 26 have been deposited in the GeneExpression Omnibus (NCBI) and are accessible online through GEO Series accession number GSE43974.LD lookupThe 1000 Genomes Project phase 3 release of variant calls was used (Feb. 20th, 2015), using 503 subjects of European ancestryPEVuZE5vdGU+PENpdGU+PEF1dGhvcj5HZW5vbWVzIFByb2plY3Q8L0F1dGhvcj48WWVhcj4yMDEy

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ADDIN EN.CITE.DATA 22. r2 between the sentinel SNPs and all other bi-allelic SNPs within the corresponding 2 Mb area was calculated using the Tabix and PLINK software package (v1.07) PEVuZE5vdGU+PENpdGU+PEF1dGhvcj5MaTwvQXV0aG9yPjxZZWFyPjIwMTE8L1llYXI+PFJlY051

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ADDIN EN.CITE.DATA 27, 28. Annotation was performed using the ANNOVAR software package ADDIN EN.CITE <EndNote><Cite><Author>Wang</Author><Year>2010</Year><RecNum>71</RecNum><DisplayText><style face="superscript">29</style></DisplayText><record><rec-number>71</rec-number><foreign-keys><key app="EN" db-id="2fxv5r22r55ep6e05xs5xxv2rae52rztt2vr" timestamp="1475036814">71</key></foreign-keys><ref-type name="Journal Article">17</ref-type><contributors><authors><author>Wang, K.</author><author>Li, M.</author><author>Hakonarson, H.</author></authors></contributors><auth-address>Center for Applied Genomics, Children&apos;s Hospital of Philadelphia, PA 19104, USA. kai@</auth-address><titles><title>ANNOVAR: functional annotation of genetic variants from high-throughput sequencing data</title><secondary-title>Nucleic Acids Res</secondary-title></titles><periodical><full-title>Nucleic Acids Res</full-title></periodical><pages>e164</pages><volume>38</volume><number>16</number><keywords><keyword>Genes</keyword><keyword>Genetic Predisposition to Disease</keyword><keyword>*Genetic Variation</keyword><keyword>Genome, Human</keyword><keyword>*Genomics</keyword><keyword>High-Throughput Screening Assays</keyword><keyword>Humans</keyword><keyword>Sequence Analysis, DNA</keyword><keyword>*Software</keyword></keywords><dates><year>2010</year><pub-dates><date>Sep</date></pub-dates></dates><isbn>1362-4962 (Electronic)&#xD;0305-1048 (Linking)</isbn><accession-num>20601685</accession-num><urls><related-urls><url> pathway analysisAll genes identified in 3 or 4 of the whole-blood eQTL resources above (Table 2), and genes containing a non-synonymous variant with r2>0.5 with the sentinel variant (Supplementary Table 13), were tested for enrichment of biological pathways and gene ontology terms using ConsensusPathDB ADDIN EN.CITE <EndNote><Cite><Author>Kamburov</Author><Year>2013</Year><RecNum>30</RecNum><DisplayText><style face="superscript">30</style></DisplayText><record><rec-number>30</rec-number><foreign-keys><key app="EN" db-id="2fxv5r22r55ep6e05xs5xxv2rae52rztt2vr" timestamp="1474361346">30</key></foreign-keys><ref-type name="Journal Article">17</ref-type><contributors><authors><author>Kamburov, A.</author><author>Stelzl, U.</author><author>Lehrach, H.</author><author>Herwig, R.</author></authors></contributors><auth-address>Department of Vertebrate Genomics, Max Planck Institute for Molecular Genetics, Ihnestrasse 63-73, 14195 Berlin, Germany. kamburov@molgen.mpg.de</auth-address><titles><title>The ConsensusPathDB interaction database: 2013 update</title><secondary-title>Nucleic Acids Res</secondary-title></titles><periodical><full-title>Nucleic Acids Res</full-title></periodical><pages>D793-800</pages><volume>41</volume><number>Database issue</number><keywords><keyword>Animals</keyword><keyword>Computer Graphics</keyword><keyword>*Databases, Genetic</keyword><keyword>*Gene Regulatory Networks</keyword><keyword>Humans</keyword><keyword>Internet</keyword><keyword>*Metabolomics</keyword><keyword>Mice</keyword><keyword>Multiprotein Complexes/genetics</keyword><keyword>*Protein Interaction Mapping</keyword><keyword>Proteins/drug effects</keyword><keyword>Proteomics</keyword><keyword>Software</keyword><keyword>Transcriptome</keyword><keyword>User-Computer Interface</keyword></keywords><dates><year>2013</year><pub-dates><date>Jan</date></pub-dates></dates><isbn>1362-4962 (Electronic)&#xD;0305-1048 (Linking)</isbn><accession-num>23143270</accession-num><urls><related-urls><url> using a FDR<5% cut-off. Enriched pathways and GO terms containing genes only implicated by a single BP-associated variant were not work analysisTo construct a functional association network, we combined two prioritized candidate gene sets into a single query gene set as (i) genes mapping to the non-synonymous SNPs (nsSNPs) in high LD (r2>0.5) with the corresponding sentinel BP associated SNP, and (ii) genes with eQTL evidence from 3 or 4 of the blood eQTL resources. Three sentinel SNPs (rs185819, rs926552 and rs805303) mapping to the HLA region on chromosome 6 were excluded from downstream analyses. The single query gene set was then used as input for the functional network analysisPEVuZE5vdGU+PENpdGU+PEF1dGhvcj5WYWV6PC9BdXRob3I+PFllYXI+MjAxNTwvWWVhcj48UmVj

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ADDIN EN.CITE.DATA 35 to identify the most relevant GO terms using the same plugin ADDIN EN.CITE <EndNote><Cite><Author>Montojo</Author><Year>2010</Year><RecNum>70</RecNum><DisplayText><style face="superscript">34</style></DisplayText><record><rec-number>70</rec-number><foreign-keys><key app="EN" db-id="2fxv5r22r55ep6e05xs5xxv2rae52rztt2vr" timestamp="1475036814">70</key></foreign-keys><ref-type name="Journal Article">17</ref-type><contributors><authors><author>Montojo, J.</author><author>Zuberi, K.</author><author>Rodriguez, H.</author><author>Kazi, F.</author><author>Wright, G.</author><author>Donaldson, S. L.</author><author>Morris, Q.</author><author>Bader, G. D.</author></authors></contributors><auth-address>Banting and Best Department of Medical Research, The Donnelly Centre, University of Toronto, 160 College Street, Toronto, ON, M5S 3E1, Canada.</auth-address><titles><title>GeneMANIA Cytoscape plugin: fast gene function predictions on the desktop</title><secondary-title>Bioinformatics</secondary-title></titles><periodical><full-title>Bioinformatics</full-title></periodical><pages>2927-8</pages><volume>26</volume><number>22</number><keywords><keyword>Algorithms</keyword><keyword>Computational Biology/*methods</keyword><keyword>Databases, Factual</keyword><keyword>Gene Regulatory Networks</keyword><keyword>Genes</keyword><keyword>*Software</keyword></keywords><dates><year>2010</year><pub-dates><date>Nov 15</date></pub-dates></dates><isbn>1367-4811 (Electronic)&#xD;1367-4803 (Linking)</isbn><accession-num>20926419</accession-num><urls><related-urls><url> Hypersensitivity overlap enrichment across tissue and cell-typesThe Functional element Overlap analysis of the Results of Genome Wide Association Study (GWAS) Experiments (Forge tool v1.1) ADDIN EN.CITE <EndNote><Cite><Author>Dunham</Author><Year>2014</Year><RecNum>31</RecNum><DisplayText><style face="superscript">36</style></DisplayText><record><rec-number>31</rec-number><foreign-keys><key app="EN" db-id="2fxv5r22r55ep6e05xs5xxv2rae52rztt2vr" timestamp="1474361630">31</key></foreign-keys><ref-type name="Journal Article">17</ref-type><contributors><authors><author>Dunham, I.</author><author>Kulesha, E.</author><author>Iotchkova, V.</author><author>Morganella, S.</author><author>Birney, E.</author></authors></contributors><titles><title>FORGE : A tool to discover cell specific enrichments of GWAS associated SNPs in regulatory regions.</title><secondary-title>BioRxiv</secondary-title></titles><periodical><full-title>BioRxiv</full-title></periodical><volume>10.1101/013045 </volume><dates><year>2014</year></dates><urls></urls></record></Cite></EndNote>36 was used to test for enrichment of overlap of BP SNPs in tissues and cell lines from the Roadmap and ENCODE projects. All 164 SNPs were entered and 143 were included in the analysis. SNPs from 9 commonly used GWAS arrays were used to select background sets of SNPs for comparison and 10,000 background repetitions were run. A Z-score threshold of >=3.39 (estimated false positive rate of 0.5%) was used to declare significance.Drug-gene interactionsGenes used for pathway and gene ontology enrichment analyses were further investigated for potential druggable or drugged targets using the drug gene interaction database (DGIdb). Known drug-gene interactions were interrogated across 15 source databases in DGIdb and include all types of interactions. The analysis performed for druggability prediction included all 9 databases exclusively inspecting expert curated data only. We also evaluate genes for known tool compounds using Chembl (ebi.ac.uk/chembl/; version 22.1).RESULTSThe stage 1 discovery meta-analysis included 150,134 individuals (Online Methods; Supplementary Tables 1-4, Supplementary Figures 1 and 2) and 7,994,604 variants with minor allele frequency (MAF) >1% and an effective sample size of at least 60% of the total (Online Methods). We identified 61 signals in the discovery analysis that were candidates for novel BP signals (P < 10-6 for any trait; Supplementary Table 5). To ensure robustness of signals, we examined BP associations in an additional 228,245 individuals from 15 independent studies for replication, including 140,886 individuals from UK Biobank PEVuZE5vdGU+PENpdGU+PEF1dGhvcj5XYXJyZW48L0F1dGhvcj48WWVhcj4yMDE3PC9ZZWFyPjxS

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ADDIN EN.CITE.DATA 19 (Supplementary Table 6 and Online Methods). We used the most significant (“sentinel”) SNP and trait for each locus in replication (61 tests). Twenty-two putatively novel association signals were initially confirmed showing significant evidence of replication in the independent stage-2 studies (P < 8.2x10-4, Bonferroni correction for 61 tests) and genome-wide significance (P < 5x10-8) in a meta-analysis across all 378,376 individuals (Online methods, Table 1, Supplementary Table 7). Of these, 14 were subsequently published in two other studies PEVuZE5vdGU+PENpdGU+PEF1dGhvcj5Ib2ZmbWFubjwvQXV0aG9yPjxZZWFyPjIwMTc8L1llYXI+

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ADDIN EN.CITE.DATA 18, 19 which presented genome-wide significant associations with evidence of replication. A further two were highlighted as putative novel signals in one of those studies ADDIN EN.CITE <EndNote><Cite><Author>Hoffmann</Author><Year>2017</Year><RecNum>82</RecNum><DisplayText><style face="superscript">18</style></DisplayText><record><rec-number>82</rec-number><foreign-keys><key app="EN" db-id="2fxv5r22r55ep6e05xs5xxv2rae52rztt2vr" timestamp="1487444910">82</key></foreign-keys><ref-type name="Journal Article">17</ref-type><contributors><authors><author>Hoffmann, T. J.</author><author>Ehret, G. B.</author><author>Nandakumar, P.</author><author>Ranatunga, D.</author><author>Schaefer, C.</author><author>Kwok, P. Y.</author><author>Iribarren, C.</author><author>Chakravarti, A.</author><author>Risch, N.</author></authors></contributors><auth-address>Department of Epidemiology and Biostatistics, University of California at San Francisco, San Francisco, California, USA.&#xD;Institute for Human Genetics, University of California at San Francisco, San Francisco, California, USA.&#xD;Center for Complex Disease Genomics, McKusick-Nathans Institute of Genetic Medicine, Baltimore, Maryland, USA.&#xD;Cardiology, Department of Specialties of Internal Medicine, University of Geneva, Geneva, Switzerland.&#xD;Kaiser Permanente Northern California Division of Research, Oakland, California, USA.</auth-address><titles><title>Genome-wide association analyses using electronic health records identify new loci influencing blood pressure variation</title><secondary-title>Nat Genet</secondary-title></titles><periodical><full-title>Nat Genet</full-title></periodical><pages>54-64</pages><volume>49</volume><number>1</number><dates><year>2017</year><pub-dates><date>Jan</date></pub-dates></dates><isbn>1546-1718 (Electronic)&#xD;1061-4036 (Linking)</isbn><accession-num>27841878</accession-num><urls><related-urls><url> but had not been confirmed by replication. In our study, we report the 6 remaining novel signals, and the 2 previously unconfirmed signals (in EBF2 and in NFKBIA), as novel signals. The 8 novel signals included 7 signals at 7 independent loci (Supplementary Figure 3) and one novel independent signal near a previously reported hit near TNXB (Online Methods, Supplementary Table 8, Supplementary Figure 4). The novel signals show both significant evidence of replication in the independent stage-2 studies (P < 8.2x10-4, Bonferroni correction for 61 tests) and genome-wide significance (P < 5x10-8) in a meta-analysis across all 378,376 individuals. The sentinel variants at all 8 signals were common (MAF>5%) and the novel secondary signal at TNXB was in high linkage-disequilibrium (r2 > 0.8) with a non-synonymous SNP. With the exception of rs9710247, which was only significant for association with DBP, all signals were significantly associated (P<0.006, Bonferroni corrected for 8 tests) with all 3 traits (Table 1 and Supplementary Table 9).We next sought to identify which genes might have expression levels that were associated with genotypes of the BP-associated variants reported in this study and others. Strong evidence of an association with expression of a specific gene may provide clues as to which gene(s) might be functionally relevant to that signal. We took the 139 BP association signals reported prior to these studies PEVuZE5vdGU+PENpdGU+PEF1dGhvcj5Ib2ZmbWFubjwvQXV0aG9yPjxZZWFyPjIwMTc8L1llYXI+

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ADDIN EN.CITE.DATA 18, 19, and 22 novel signals of association identified and confirmed in this study and two contemporaneous studies ZW50IG9mIE1lZGljYWwgU2NpZW5jZSBhbmQgQ2FyZGlvcmVuYWwgTWVkaWNpbmUsIFlva29oYW1h

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ADDIN EN.CITE.DATA 3-19, 24 (Supplementary Table 10), and searched for evidence of association with gene expression in whole-blood (four studies, total n=12,607; Online Methods) and in kidney tissue (n=134, the largest kidney eQTL resource currently available). Although of unclear direct relevance to BP, whole-blood was studied due to the availability of large data sets enabling a powerful assessment of expression patterns that are likely present across multiple cell and tissue types. Similarly, circulating blood cells have been used for ion transport experiments in the past and altered ion transport levels in erythrocytes were linked to hypertension. ADDIN EN.CITE <EndNote><Cite><Author>Trevisan</Author><Year>1983</Year><RecNum>83</RecNum><DisplayText><style face="superscript">37</style></DisplayText><record><rec-number>83</rec-number><foreign-keys><key app="EN" db-id="2fxv5r22r55ep6e05xs5xxv2rae52rztt2vr" timestamp="1493628178">83</key></foreign-keys><ref-type name="Journal Article">17</ref-type><contributors><authors><author>Trevisan, M.</author><author>Ostrow, D.</author><author>Cooper, R.</author><author>Liu, K.</author><author>Sparks, S.</author><author>Okonek, A.</author><author>Stevens, E.</author><author>Marquardt, J.</author><author>Stamler, J.</author></authors></contributors><titles><title>Abnormal red blood cell ion transport and hypertension. The People&apos;s Gas Company study</title><secondary-title>Hypertension</secondary-title></titles><periodical><full-title>Hypertension</full-title><abbr-1>Hypertension</abbr-1></periodical><pages>363-7</pages><volume>5</volume><number>3</number><keywords><keyword>Adult</keyword><keyword>Age Factors</keyword><keyword>Biological Transport, Active/drug effects</keyword><keyword>Blood Pressure</keyword><keyword>Body Weight</keyword><keyword>Erythrocytes/*metabolism</keyword><keyword>Humans</keyword><keyword>Hypertension/*metabolism</keyword><keyword>Ion Exchange</keyword><keyword>Lithium/metabolism</keyword><keyword>Male</keyword><keyword>Middle Aged</keyword><keyword>Potassium/blood</keyword><keyword>Sodium/blood/metabolism</keyword></keywords><dates><year>1983</year><pub-dates><date>May-Jun</date></pub-dates></dates><isbn>0194-911X (Print)&#xD;0194-911X (Linking)</isbn><accession-num>6840823</accession-num><urls><related-urls><url> Kidney was chosen because of the many renal pathways that regulate BP and outstanding questions about the relevance of kidney pathways to the genetic component of BP regulation in the general population TWVkaWNpbmUsIEVyYXNtdXMgTUMsIFJvdHRlcmRhbSwgdGhlIE5ldGhlcmxhbmRzLiYjeEQ7RGVw

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ADDIN EN.CITE.DATA 3, 15. Expression quantitative trait loci (eQTL) signals were filtered by false discovery rate (FDR<5%) and we examined cis (within 1Mb) associations only (Online methods and Supporting Information).The four blood eQTL data sets were NESDA-NTR PEVuZE5vdGU+PENpdGU+PEF1dGhvcj5XcmlnaHQ8L0F1dGhvcj48WWVhcj4yMDE0PC9ZZWFyPjxS

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ADDIN EN.CITE.DATA 15, the BIOS resource ADDIN EN.CITE <EndNote><Cite><Author>Zhernakova</Author><Year>2015</Year><RecNum>27</RecNum><DisplayText><style face="superscript">40</style></DisplayText><record><rec-number>27</rec-number><foreign-keys><key app="EN" db-id="2fxv5r22r55ep6e05xs5xxv2rae52rztt2vr" timestamp="1474021949">27</key></foreign-keys><ref-type name="Journal Article">17</ref-type><contributors><authors><author>Zhernakova, D.</author><author>Deelen, P.</author><author>Vermaat, M.</author><author>van Iterson, M.</author><author>van Galen, M.</author></authors></contributors><titles><title>Hypothesis-free identification of modulators of genetic risk factors</title><secondary-title>BioRxiv</secondary-title></titles><periodical><full-title>BioRxiv</full-title></periodical><pages>dx.10.1101/033217</pages><dates><year>2015</year></dates><urls></urls></record></Cite></EndNote>40 and GTEx ADDIN EN.CITE <EndNote><Cite><Author>Consortium</Author><Year>2015</Year><RecNum>28</RecNum><DisplayText><style face="superscript">25</style></DisplayText><record><rec-number>28</rec-number><foreign-keys><key app="EN" db-id="2fxv5r22r55ep6e05xs5xxv2rae52rztt2vr" timestamp="1474022265">28</key></foreign-keys><ref-type name="Journal Article">17</ref-type><contributors><authors><author>G. TEx Consortium</author></authors></contributors><titles><title>Human genomics. The Genotype-Tissue Expression (GTEx) pilot analysis: multitissue gene regulation in humans</title><secondary-title>Science</secondary-title></titles><periodical><full-title>Science</full-title></periodical><pages>648-60</pages><volume>348</volume><number>6235</number><keywords><keyword>Alleles</keyword><keyword>Blood Pressure/genetics</keyword><keyword>Disease/*genetics</keyword><keyword>GTPase-Activating Proteins/genetics</keyword><keyword>*Gene Expression Regulation</keyword><keyword>Gene Regulatory Networks</keyword><keyword>*Genetic Variation</keyword><keyword>Genome, Human/*genetics</keyword><keyword>Genome-Wide Association Study</keyword><keyword>Genotype</keyword><keyword>Humans</keyword><keyword>Multigene Family</keyword><keyword>Organ Specificity/genetics</keyword><keyword>Pilot Projects</keyword><keyword>*Quantitative Trait Loci</keyword><keyword>RNA Splicing</keyword><keyword>RNA, Untranslated/genetics</keyword><keyword>Sequence Analysis, RNA</keyword><keyword>Tibial Arteries/metabolism</keyword><keyword>*Transcriptome</keyword></keywords><dates><year>2015</year><pub-dates><date>May 8</date></pub-dates></dates><isbn>1095-9203 (Electronic)&#xD;0036-8075 (Linking)</isbn><accession-num>25954001</accession-num><urls><related-urls><url> (Online Methods and Supporting Information). The BIOS resource (n=2,116) has not previously been utilized in the analysis of BP associations, findings from NESDA-NTR and SABRe have been reported for a subset of the previously published signals IEVuZ2xhbmQgQ2VudHJlIGZvciBFbnZpcm9ubWVudCBhbmQgSGVhbHRoLCBTY2hvb2wgb2YgUHVi

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ADDIN EN.CITE.DATA 16, 17. For a total of 369 genes, gene-expression was associated with the BP SNP in one or more of the 4 blood datasets at experiment-wide significance (Supplementary Table 11). This included 14 genes for 6 of the 8 novel signals. For 110 genes, we found eQTL evidence in 2 out of 4 datasets (Figure 1), including 4 genes for 2 of the novel signals; EIF4B and TNS2 for rs73099903 and MAP3K10 and PLD3 for rs9710247. SNP rs73099903 was in strong linkage disequilibrium (LD r2>0.9) with the SNP most strongly associated with TNS2 expression in the BIOS resource. TNS2 encodes a tensin focal adhesion molecule and may have a role in renal function ADDIN EN.CITE <EndNote><Cite><Author>Marusugi</Author><Year>2016</Year><RecNum>83</RecNum><DisplayText><style face="superscript">41</style></DisplayText><record><rec-number>83</rec-number><foreign-keys><key app="EN" db-id="2fxv5r22r55ep6e05xs5xxv2rae52rztt2vr" timestamp="1487509991">83</key></foreign-keys><ref-type name="Journal Article">17</ref-type><contributors><authors><author>Marusugi, K.</author><author>Nakano, K.</author><author>Sasaki, H.</author><author>Kimura, J.</author><author>Yanobu-Takanashi, R.</author><author>Okamura, T.</author><author>Sasaki, N.</author></authors></contributors><auth-address>Laboratory of Laboratory Animal Science and Medicine, School of Veterinary Medicine, Kitasato University, Towada, Aomori 034-8628, Japan.</auth-address><titles><title>Functional validation of tensin2 SH2-PTB domain by CRISPR/Cas9-mediated genome editing</title><secondary-title>J Vet Med Sci</secondary-title></titles><periodical><full-title>J Vet Med Sci</full-title></periodical><pages>1413-1420</pages><volume>78</volume><number>9</number><dates><year>2016</year><pub-dates><date>Oct 01</date></pub-dates></dates><isbn>1347-7439 (Electronic)&#xD;0916-7250 (Linking)</isbn><accession-num>27246398</accession-num><urls><related-urls><url> 48 genes, we found evidence in 3 out of the 4 resources (Table 2), suggesting robustness of the SNP-gene expression correlation signal and highlighting those genes as potential candidates in genetic BP regulation. Of the 48 genes, 28 have not previously been described in eQTL analyses using BP associated SNPs and all were correlated with previously reported BP association signals.In the kidney dataset (TransplantLines) PEVuZE5vdGU+PENpdGU+PEF1dGhvcj5EYW1tYW48L0F1dGhvcj48WWVhcj4yMDE1PC9ZZWFyPjxS

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ADDIN EN.CITE.DATA 26, there was association of gene expression and genotype for nine SNPs and 13 genes (Table 2, Figure 1 and Supplementary Table 12). Nine of the SNP-gene expression associations were also observed in the whole-blood eQTL datasets, suggesting that those signals may not be unique to the kidney. We report three signals that were unique to the kidney and not previously reported (C4orf34, HIP2 and ASIC1) and confirm a previously reported kidney eQTL signal for an anti-sense RNA for PSMD5 aWNpbmUsIEVyYXNtdXMgTUMsIFJvdHRlcmRhbSwgdGhlIE5ldGhlcmxhbmRzLiYjeEQ7RGVwYXJ0

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RW5kTm90ZT4A

ADDIN EN.CITE.DATA 42. The comparatively small number of signals using kidney tissue (Table 2 and Figure 1) compared to whole-blood could be due to the small sample size. Complete GTEx results are in Supplementary Table 13.For genes implicated by eQTL information from whole-blood, we tested for enrichment of biological pathways and gene ontologies (Online Methods). We noted enrichment of the 48 genes implicated by 3 or 4 blood eQTL resources, Table 2, and a further 53 genes containing a non-synonymous variant with r2 > 0.5 with the top SNP (Supplementary Table 14), in pathways and ontology terms related to actin and striated muscle (Supplementary Tables 15 and 16, Online Methods). Network analysis using the same genes highlighted further GO terms relating to muscle function, particularly cardiac muscle (Online Methods, Supplementary Table 17). We tested the overlap of 161 non-HLA BP associated variants with DNase Hypersensitivity sites identified in the Roadmap and ENCODE cell lines (Online Methods) and identified an overall enrichment in multiple cell and tissue types including heart, kidney and smooth muscle (Supplementary Figure 5).We next investigated these genes for potential suitability as drug targets (druggability), known tool compounds and clinically approved drugs using the drug gene interaction database (DGIdb) PEVuZE5vdGU+PENpdGU+PEF1dGhvcj5XYWduZXI8L0F1dGhvcj48WWVhcj4yMDE2PC9ZZWFyPjxS

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ADDIN EN.CITE.DATA 43 (Supplementary Table 18). Twelve genes had known drugs, including four genes with known antihypertensive drugs. We noted that drugs modulating all but one of the 12 drugged targets had a reported influence on blood pressure, either as a primary antihypertensive indication or as a reported side effect of raised blood pressure. Twenty additional genes were predicted druggable, among these 7 genes have known small molecule tool modulators, based on a query of the Chembl database (ebi.ac.uk/chembldb/; version 22.1). DISCUSSIONEnhanced discovery of BP loci increases the potential targets for therapeutic advances. After major advances in the number of BP loci known over the last years and months, we report 8 novel signals that implicate 5 regions of the genome not previously connected to blood pressure regulation. Six of the 8 novel signals we report had not previously been reported. Two signals (in EBF2 and NFKBIA) have been suggested previously but without evidence for replication ADDIN EN.CITE <EndNote><Cite><Author>Hoffmann</Author><Year>2017</Year><RecNum>82</RecNum><DisplayText><style face="superscript">18</style></DisplayText><record><rec-number>82</rec-number><foreign-keys><key app="EN" db-id="2fxv5r22r55ep6e05xs5xxv2rae52rztt2vr" timestamp="1487444910">82</key></foreign-keys><ref-type name="Journal Article">17</ref-type><contributors><authors><author>Hoffmann, T. J.</author><author>Ehret, G. B.</author><author>Nandakumar, P.</author><author>Ranatunga, D.</author><author>Schaefer, C.</author><author>Kwok, P. Y.</author><author>Iribarren, C.</author><author>Chakravarti, A.</author><author>Risch, N.</author></authors></contributors><auth-address>Department of Epidemiology and Biostatistics, University of California at San Francisco, San Francisco, California, USA.&#xD;Institute for Human Genetics, University of California at San Francisco, San Francisco, California, USA.&#xD;Center for Complex Disease Genomics, McKusick-Nathans Institute of Genetic Medicine, Baltimore, Maryland, USA.&#xD;Cardiology, Department of Specialties of Internal Medicine, University of Geneva, Geneva, Switzerland.&#xD;Kaiser Permanente Northern California Division of Research, Oakland, California, USA.</auth-address><titles><title>Genome-wide association analyses using electronic health records identify new loci influencing blood pressure variation</title><secondary-title>Nat Genet</secondary-title></titles><periodical><full-title>Nat Genet</full-title></periodical><pages>54-64</pages><volume>49</volume><number>1</number><dates><year>2017</year><pub-dates><date>Jan</date></pub-dates></dates><isbn>1546-1718 (Electronic)&#xD;1061-4036 (Linking)</isbn><accession-num>27841878</accession-num><urls><related-urls><url>. For these two signals we present, for the first time, stringent evidence of replication, confirming their relevance to blood pressure genetics.The path from signal to genes is the essential next step towards realizing the therapeutic potential of a genetic locus and understanding the mechanisms of BP regulation. We have used several large eQTL resources as a first step to realize this objective. As expected, we observed that even across eQTL studies of the same tissue, there is limited overlap in experiment-wide significant signals suggesting either biologic variability (differences in the characteristics of the samples or in the methods for extraction and processing of mRNA in each of the studies), technology-specific differences in coverage of genes (use RNAseq data for the BIOS blood dataset and microarray-based expression levels for the kidney and other blood datasets), or the possibility of false positive results despite stringent within-experiment significance thresholds. We were unable to distinguish these scenarios using the data available to us but by selecting genes that were significant in at least three resources, and therefore robust to these differences, we identified 48 genes as candidates for further study. These results are limited by the availability of large eQTL resources for whole-blood only, which precludes well-powered comparisons across tissue types, particularly as the origin of blood pressure control is unlikely to be located in the blood. Enrichment and pathway analyses using these genes, and genes containing a correlated functional variant, highlight the potential relevance of muscular tissue and pathways, compatible with a vascular and cardiac origin of BP genetics, extending previous evidence aWNpbmUsIEVyYXNtdXMgTUMsIFJvdHRlcmRhbSwgdGhlIE5ldGhlcmxhbmRzLiYjeEQ7RGVwYXJ0

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ADDIN EN.CITE.DATA 15. We identify a number of drugged targets in the pathways identified, including four existing hypertension targets. Other drugs identified are not suitable candidates for repositioning to hypertension, as most were reported in adverse events to raise blood pressure, however the targets would be valid for investigation using a reverse mechanism, e.g. agonism in place of inhibition. We also identified seven genes with small molecule tool modulators (mainly inhibitory or binding). These molecules and targets might be suitable candidates for further investigation to build a target validation case to support clinical investigation in hypertension.Amongst the genes implicated in our eQTL analyses were several for which there is already some evidence that they are relevant to blood pressure regulation. The intronic SNP rs10926988 was independently associated with expression of SDCCAG8 in all four whole-blood resources. Rare mutations in SDCCAG8 cause Bardet-Biedl syndrome, which features hypertension. Expression levels of MYBPC3 were correlated with rs7103648aWNpbmUsIEVyYXNtdXMgTUMsIFJvdHRlcmRhbSwgdGhlIE5ldGhlcmxhbmRzLiYjeEQ7RGVwYXJ0

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ADDIN EN.CITE.DATA 44This study has several limitations: Given the nature of statistical power for genome-wide association analyses, the sample size is limited, even though this is one of the largest efforts in BP GWAS undertaken so far. The study would clearly have benefited from the availability of larger eQTL resources on multiple tissues in sample sizes even larger than those available today. Our analyses were limited to cis-signals and future analyses, with larger sample sizes, might also consider trans-signals.In summary, our study reports novel BP association signals and reports new candidate BP genes, contributing to the transition from variants to genes to explain BP variation.DISCLOSURESThe authors declare competing financial interests (see corresponding section in the Supporting Information).SOURCES OF FUNDING: See end of the manuscript.NOTE: Online data supplements are available in the online version of the paper.ACKNOWLEDGEMENTSWe thank all the study participants of this study for their contributions. Detailed acknowledgment of funding sources is provided in the Supporting Information.REFERENCES ADDIN EN.REFLIST 1.Nelson MR, Tipney H, Painter JL, Shen J, Nicoletti P, Shen Y, Floratos A, Sham PC, Li MJ, Wang J, Cardon LR, Whittaker JC, Sanseau P. The support of human genetic evidence for approved drug indications. 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Gene. 2015;573:188-197NOVELTY AND SIGNIFICANCEWhat is New: The root origin of hypertension and hence blood pressure variability in the population remains unclear. This study adds data to explain the genetic basis of blood pressure variability and identifies genes likely active in blood pressure regulating pathways.What Is Relevant: The results are of relevance for scientists, clinicians, and pharmacologists interested in hypertension. The BP loci and the BP genes identified constitute new leads for the understanding of BP pathogenesis and possibly therapeutic innovation.Summary: Using 1000 Genomes Project-based imputation in 150,134 European ancestry and independent replication in a further 228,245 individuals we contribute 8 replicated blood pressure loci to the collection of loci currently known. Using these and previous data, 48 BP genes are identified for priority follow-up.FIGURE LEGENDSFigure 1: Overlap of eQTL evidence from four whole-blood and one kidney resourceThe figure indicates overlap of evidence for eQTLs from four whole-blood studies (SABRe, NESDA-NTR, BIOS, and GTEx) and from one kidney resource (TransplantLines). Every colored line indicates that this gene was analysis-wide significant in a given resource (see Online Methods). Only genes identified by at least two resources are shown. The genes are sorted by genomic position on the y-axis.FIGURESFigure 11485900125730000Table 1. Novel genome-wide significant signals of associationResults from stage 1 and stage 2, and the meta-analysis of stage 1 and stage 2, for all novel genome-wide significant signals of association. P values of association for all 3 traits from a meta-analysis of stages 1 and 2 are also presented. Genome-wide significant P values (P<5x10-8) are in bold. Abbreviations: CAF: coded allele frequency se: standard error, Neff: effective sample size. #Novel signal at previously reported locus. 1For intragenic variants the nearest genes are listed, all other variants are intronic unless indicated otherwise; ns= non-synonymous, s=synonymous, UTR= Untranslated Region. Results from proxy SNPs are indicated by (proxy); rs848309 was a proxy SNP for rs1048238 and rs10926988 was a proxy SNP for chr1:243458005:I.Results for most significant traitStage 1 + stage 2 meta-analysis P values for all traitsStage 1Stage 2Stage 1+ stage 2Variant ID (noncoded/coded allele) chr:position, Nearest gene(s)(type1)CAFBeta (se)P valueNeffBeta (se)P valueNeffBeta (se)P valueNeffSBPDBPPPSBPrs1048238 (C/T)1:16341649, HSPB7 (3’UTR)0.5710.366(0.074)8.09E-07140299NANANANANANANANANArs848309(proxy) (T/C)1:163084470.5670.347(0.072)1.70E-061467550.347(0.071)9.10E-071404620.347(0.051)7.07E-122872177.07E-121.07E-105.48E-06#rs185819 (T/C)6:32,050,067, TNXB (ns)0.5130.534(0.073)1.93E-131423970.277(0.053)1.49E-072217480.365(0.043)1.04E-173641441.04E-172.24E-118.50E-15rs6557876 (C/T)8:25,900,675, EBF20.252-0.411(0.084)8.50E-07143653-0.350(0.060)5.66E-09225803-0.371(0.049)2.85E-143694572.85E-142.50E-101.51E-08rs35783704 (G/A)8:105,966,258, LRP12/ZFPM20.109-0.609(0.121)4.96E-07133924-0.310(0.089)4.78E-04215528-0.414(0.072)7.08E-093494527.08E-091.60E-062.92E-07rs73099903 (C/T)12:53,440,779, LOC2833350.0740.768(0.143)8.05E-081360640.396(0.098)5.32E-052072530.515(0.081)1.95E-103433181.95E-104.53E-065.46E-08rs8904 (G/A)14:35,871,217, NFKBIA (3’ UTR)0.3750.377(0.076)6.76E-071404240.278(0.054)2.31E-072247710.311(0.044)1.31E-123651951.31E-121.13E-043.44E-12rs57927100 (C/G)17:75,317,300, SEPT90.258-0.489(0.086)1.10E-08136624-0.220(0.061)3.12E-04210563-0.310(0.050)4.04E-103471884.04E-101.16E-101.81E-05DBPrs9710247 (A/G)19:40,760,449, AKT20.4470.252(0.051)8.11E-071096950.129(0.032)5.76E-051983320.164(0.027)1.61E-093080283.82E-021.61E-095.03E-01Table 2: BP associated SNPs associated with expression of the same gene across 4 or 3 independent whole-blood eQTL resources and the kidney resource. Signals of association of SNP genotype and gene expression in other non-blood tissues in GTEx and in kidney are also indicated. Blood dataset order: (i) SABRe, (ii) NESDA-NTR, (iii) BIOS, (iv) GTEx (whole-blood). Top eQTL: Top GWAS SNP is top eQTL SNP (or in high LD, r2>0.9, with top eQTL SNP) in at least one data set. eQTL signal previously reported: Genes for which eQTL signals have been previously reported for that sentinel SNPdXJnaCwgVUsuJiN4RDtRdWVlbnNsYW5kIEJyYWluIEluc3RpdHV0ZSwgVW5pdmVyc2l0eSBvZiBR

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ZE5vdGU+

ADDIN EN.CITE.DATA 15-17. For full list, see Supplementary Table 12.Sentinel SNPChrPositionGeneBlood data sets Top eQTLSignal in other tissue(s) in GTExSignal in kidneyeQTL signal previously reportedSignal in 4 whole-blood eQTL resourcesrs17367504111862778CLCN6YYYYYYrs21691371204497913MDM4YYYYYYYrs109269881243483279SDCCAG8YYYYYrs319690347927484MAP4YYYYYYYrs125218685131784393SLC22A5YYYYYrs9001451113293905ARNTLYYYYYYrs106010512123806219CDK2AP1YYYYYYYrs13789421575077367SCAMP2YYYYrs11264641689704365CHMP1AYYYYYYrs11264641689704365FANCAYYYYYrs129464541743208121DCAKDYYYYYYYSignal in 3 (out of 4) whole-blood eQTL resourcesrs17367504111862778MTHFRYYYNYYrs871524138411445FHL3NYYYYrs871524138411445SF3A3NYYYYrs4660293140028180PABPC4YYYNYYYrs67494472169041386STK39YYYNYrs347591311290122ATG7YYYNYrs319690347927484ZNF589YYNYYrs125218685131784393SLC22A4YYYNYrs1563788643308363CRIP3YYYNYYrs10943605679655477PHIPYYYNYYYrs47281427128573967IRF5NYYYYYYrs47281427128573967TNPO3YYYNYrs2898290811433909BLKYYYNYrs2898290811433909FAM167ANYYYYrs2898290811433909FDFT1YYYNYrs20715188120435812NOVYYYNYrs76452347935906471TPM2YYYNrs107601179123586737MEGF9YYYNYYrs44942501096563757HELLSYYYNYrs1119154810104846178NT5C2YYYNYrs661348111905292TNNT3NYYYYrs2649044119763969SBF2YYYNrs2649044119763969SWAP70YYYNYY?rs71292201110350538ADMYYYNYrs71036481147461783MYBPC3YYYNrs37413781165408937CTSWYYYNrs73029811250537815LIMA1YYYNYrs73029811250537815ATF1YYNYYrs10364771548914926FBN1YNYYrs13789421575077367CSKYYYNYYYrs13789421575077367MPINYYYYrs13789421575077367ULK3YNYYYYrs129464541743208121NMT1YYYNYrs23041301919789528GATAD2AYYYNrs8671862033764554EIF6NYYYYrs60952412047308798PREX1YYYNrs93061602145107562RRP1BYNYYYYCONTRIBUTIONS / ACKNOWLEDGMENTSAUTHOR CONTRIBUTIONSSecondary analysesDesign of secondary analyses: L.V.W., G.B.E, M.J.C., H.Snieder, M.D.T , R.Joehanes, A.V., R.Jansen, A.V., J.K., P.O.R., A.P.M., C.P.C. Computation of secondary analysis: L.V.W., G.B.E., A.P.M., M.E., T.B., L.Lin, R.Joehanes, A.V., P.J.v.d.M., R.Jansen, C.P.C.DiscoveryWGHS : Study phenotyping: P.M.R. Genotyping or analysis: D.I.C., L.M.R. Study PI: D.I.C., P.M.R. RS : Study phenotyping: G.C.V. Genotyping or analysis: G.C.V., A.G.U. Study PI: O.H.F., A.Hofman, A.G.U. NTR : Study phenotyping: E.J.d.G., G.W. Genotyping or analysis: J.J.H., E.J.d.G., G.W. Study PI: D.I.B., E.J.d.G. STR : Study phenotyping: E.I. Genotyping or analysis: R.J.S., M.Fr?nberg Study PI: E.I., A.Hamsten EGCUT : Genotyping or analysis: T.E. Study PI: A.Metspalu ARIC : Genotyping or analysis: D.E.A., A.C.M., P.N. Study PI: A.Chakravarti FHS : Study phenotyping: D.L. Genotyping or analysis: S.J.H. Study PI: D.L. MESA : Study phenotyping: J.I.R. Genotyping or analysis: W.P., X.G., J.I.R., J.Y. Study PI: W.P. B58C : Study phenotyping: D.P.S. Genotyping or analysis: D.P.S. Study PI: D.P.S. COLAUS : Study phenotyping: P.V. Genotyping or analysis: M.Bochud, Z.K. Study PI: P.V. PROSPER : Study phenotyping: J.W.J., D.J.S. Genotyping or analysis: S.Trompet, J.D. Study PI: J.W.J. BHS : Study phenotyping: A.James Genotyping or analysis: N.Shrine, J.H., J.B. SHIP : Study phenotyping: M.D. Genotyping or analysis: A.T., M.D., U.V. Study PI: R.R. KORA S4 : Genotyping or analysis: J.S.R. Study PI: A.Peters CHS : Study phenotyping: B.M.P. Genotyping or analysis: J.C.B., K.R., K.D.T. Study PI: B.M.P. AGES-Reykjavik : Genotyping or analysis: A.V.S. Study PI: V.Gudnason, T.B.H., L.J.L. ERF : Study phenotyping: C.M.v.D., B.A.O. Genotyping or analysis: N.A. Study PI: C.M.v.D., B.A.O. NESDA : Study phenotyping: B.W.J.H.P. Genotyping or analysis: I.M.N., Y.M. Study PI: H.Snieder, B.W.J.H.P. YFS : Study phenotyping: T.L., M.K., O.T.R. Genotyping or analysis: T.L., L.P.L., M.K., O.T.R. Study PI: T.L., M.K., O.T.R. EPIC : Genotyping or analysis: N.J.W. Study PI: J.H.Z. ASPS : Study phenotyping: R.Schmidt Genotyping or analysis: H.Schmidt, E.H., Y.S., R.Schmidt Study PI: H.Schmidt, R.Schmidt ORCADES : Study phenotyping: J.F.W., H.C., S.W. Genotyping or analysis: J.F.W., P.K.J., S.W. Study PI: J.F.W. FINRISK (COROGENE_CTRL) : Study phenotyping: P.J. Genotyping or analysis: K.K., A.P.S. Study PI: M.P., P.J. INGI-VB : Study phenotyping: C.F.S. Genotyping or analysis: M.T., C.M.B., C.F.S. Study PI: D.T. FINRISK_PREDICT_CVD : Study phenotyping: V.S., A.S.H. Study PI: V.S., A.Palotie, S.R. TRAILS : Study phenotyping: H.R. Genotyping or analysis: P.J.v.d.M. Study PI: C.A.H., A.J.O. PROCARDIS : Study phenotyping: A.G. Genotyping or analysis: A.G. Study PI: H.W., M.Farrall HABC : Study phenotyping: Y.Liu, T.B.H. Genotyping or analysis: M.A.N. Study PI: Y.Liu, T.B.H. KORA S3 : Study phenotyping: C.G. Genotyping or analysis: S.S., C.G., E.O. Study PI: M.Laan INGI-FVG : Genotyping or analysis: D.V., M.Brumat, M.Cocca Study PI: P.G. Fenland : Study phenotyping: R.A.S., J.a.L., C.L., N.J.W. Genotyping or analysis: R.A.S., J.a.L., C.L., N.J.W. Study PI: R.A.S., C.L., N.J.W. MICROS : Genotyping or analysis: A.A.H., F.D.G.M., A.S.P. Study PI: F.D.G.M., P.P.P. HTO : Study phenotyping: B.D.K. Genotyping or analysis: B.D.K., K.L.A., C.Mamasoula Study PI: B.D.K., H.J.C. MIGEN : Study phenotyping: R.E., J.Marrugat, S.Kathiresan, D.S. Genotyping or analysis: R.E., S.Kathiresan, D.S. Study PI: S.Kathiresan ULSAM : Study phenotyping: V.Giedraitis, E.I. Genotyping or analysis: A.P.M., A.Mahajan Study PI: A.P.M., V.Giedraitis, E.I. Cilento study : Study phenotyping: R.Sorice Genotyping or analysis: D.R., T.Nutile Study PI: M.Ciullo LBC1936 : Study phenotyping: I.J.D., A.J.G. Genotyping or analysis: L.M.L., G.D., A.J.G. Study PI: I.J.D. H2000_CTRL : Study phenotyping: T.Niiranen Study PI: P.K., A.Jula, S.Koskinen NSPHS : Genotyping or analysis: S.E., ?.J. Study PI: U.G. FUSION : Genotyping or analysis: A.U.J. Study PI: J.T., M.Boehnke, F.C. GRAPHIC : Study phenotyping: N.J.S., P.S.B., M.D.T. Genotyping or analysis: C.P.N., P.S.B., M.D.T. Study PI: N.J.S. CROATIA_Vis : Study phenotyping: I.R. Genotyping or analysis: V.V., J.E.H. Study PI: V.V., I.R. PIVUS : Study phenotyping: L.Lind, J.S. Genotyping or analysis: C.M.L., A.Mahajan Study PI: C.M.L., L.Lind, J.S. LOLIPOP : Study phenotyping: J.S.K., J.C.C. Genotyping or analysis: J.S.K., W.Z., J.C.C., B.L. Study PI: J.S.K., J.C.C. CROATIA_Korcula : Genotyping or analysis: C.H., J.Marten Study PI: C.H., A.F.W. INGI-CARL : Study phenotyping: G.G. Genotyping or analysis: I.G., A.Morgan, A.R. LBC1921 : Study phenotyping: J.M.S., A.Pattie Genotyping or analysis: J.M.S., S.E.H., D.C.M.L., A.Pattie Study PI: J.M.S. CROATIA_SPLIT : Study phenotyping: O.P., I.K. Genotyping or analysis: O.P., T.Z. Study PI: O.P. BioMe (formerly IPM) : Genotyping or analysis: Y.Lu Study PI: R.J.F.L., E.P.B. ReplicationUKB-BP : Genotyping or analysis: H.R.W., M.R.B., C.P.C., E.E., H.G., B.M., M.R., I.T. Study PI: P.E., M.J.C. GoDARTS : Study phenotyping: C.N.A.P., A.S.F.D. Genotyping or analysis: C.N.A.P., N.Shah Study PI: C.N.A.P., A.D.M. Lifelines : Study phenotyping: M.H.d.B. Genotyping or analysis: M.S. Study PI: P.v.d.H. TwinsUK : Study phenotyping: C.Menni Genotyping or analysis: M.M., C.Menni Study PI: T.D.S. Airwave Health Monitoring Study : Genotyping or analysis: A.C.V., E.E., H.G., I.T. Study PI: E.E. The UK Household Longitudinal Study (UKHLS) : Genotyping or analysis: B.P.P. Study PI: E.Z. Generation Scotland (GS:SFHS) : Study phenotyping: S.P. Genotyping or analysis: C.H., A.Campbell JUPITER : Study phenotyping: P.M.R. Genotyping or analysis: D.I.C., L.M.R., F.G., P.M.R. Study PI: D.I.C., P.M.R. NEO : Study phenotyping: R.d.M. Genotyping or analysis: D.O.M.K., R.L.G. Study PI: R.d.M. Three City-Dijon : Study phenotyping: S.D., C.T. Genotyping or analysis: G.C. Study PI: S.D., C.T. ASCOT-UK : Study phenotyping: P.S., N.P. Genotyping or analysis: P.B.M., H.R.W. Study PI: P.B.M., P.S., N.P., M.J.C. ASCOT-SC : Study phenotyping: S.Thom, M.J.C. Genotyping or analysis: D.C.S., A.S., H.R.W., P.B.M. Study PI: S.Thom, M.J.C., P.B.M. Hunter Community Study : Study phenotyping: R.Scott Genotyping or analysis: C.O., E.G.H. Study PI: A.John GAPP : Study phenotyping: D.C. Genotyping or analysis: D.C., S.Thériault, G.P. Study PI: D.C. BRIGHT : Study phenotyping: M.Brown, J.C. Genotyping or analysis: M.Farrall, P.B.M., H.R.W. Study PI: M.Brown, J.C., M.Farrall, P.B.M., M.J.C. Resources for secondary analyseseQTL NESDA NTR : Design of secondary analysis: R.Jansen Computation of secondary analysis: D.I.B., R.Jansen, B.W.J.H.P. Study PI: D.I.B., B.W.J.H.P. eQTL kidney : Study phenotyping: J.J.D., M.A.S. Genotyping or analysis: P.J.v.d.M. Study PI: H.Snieder eQTL BIOS : Design of secondary analysis: R.Jansen Computation of secondary analysis: R.Jansen Study PI: R.Jansen SABRe : Study phenotyping: Y.D., P.J.M., Q.T.N. Genotyping or analysis: R.Joehanes Design of secondary analysis: D.L. Study PI: D.L. ICBP-Steering CommitteeG.A., M.J.C., A.Chakravarti, D.I.C., G.B.E., P.E., T.F., M.R.J., A.D.J., M.Larson, D.L., A.P.M., P.B.M., C.N.C., P.O.R., W.P., B.M.P., K.R., A.V.S., H.Snieder, M.D.T., C.M.v.D., L.V.W., H.R.W.ACKNOWLEDGMENTSThis research used the ALICE and SPECTRE High Performance Computing Facilities at the University of Leicester. G.B.E is supported by Geneva University Hospitals, Geneva University, de Reuter Foundation, the Swiss National Foundation project FN 33CM30-124087, and the “Fondation pour Recherches Médicales”, Geneva.Airwave: We thank all participants of the Airwave Health Monitoring Study. The study is funded by the UK Home Office, (Grant number 780-TETRA) with additional support from the National Institute for Health Research Imperial College Health Care NHS Trust and Imperial College Biomedical Research Centre.ARIC: The Atherosclerosis Risk in Communities Study is carried out as a collaborative study supported by National Heart, Lung, and Blood Institute contracts (HHSN268201100005C, HHSN268201100006C, HHSN268201100007C, HHSN268201100008C, HHSN268201100009C, HHSN268201100010C, HHSN268201100011C, and HHSN268201100012C), R01HL087641, R01HL59367 and R01HL086694; National Human Genome Research Institute contract U01HG004402; and National Institutes of Health contract HHSN268200625226C. Funding support for the Genetic Epidemiology of Causal Variants Across the Life Course (CALiCo) program was provided through the NHGRI PAGE program (U01 HG007416). The authors thank the staff and participants of the ARIC study for their important contributions. The authors thank the staff and participants of the ARIC study for their important contributions. ASCOT: This work was supported by Pfizer, New York, NY, USA, for the ASCOT study and the collection of the ASCOT DNA repository; by Servier Research Group, Paris, France; and by Leo Laboratories, Copenhagen, Denmark. We thank all ASCOT trial participants, physicians, nurses, and practices in the participating countries for their important contribution to the study. In particular we thank Clare Muckian and David Toomey for their help in DNA extraction, storage, and handling. This work forms part of the research programme of the NIHR Cardiovascular Biomedical Research Unit at Barts ASPS: The research reported in this article was funded by the Austrian Science Fond (FWF) grant number P20545-P05 and P13180. The Medical University of Graz supports the databank of the ASPS. The authors thank the staff and the participants of the ASPS for their valuable contributions. The authors thank Birgit Reinhart for her long-term administrative commitment and Ing Johann Semmler for the technical assistance at creating the DNA bank.?BRIGHT: This work was supported by the Medical Research Council of Great Britain (grant number G9521010D); and by the British Heart Foundation (grant number PG/02/128). The BRIGHT study is extremely grateful to all the patients who participated in the study and the BRIGHT nursing team. This work forms part of the research programme of the NIHR Cardiovascular Biomedical Research Unit at Barts. B58C: We acknowledge use of phenotype and genotype data from the British 1958 Birth Cohort DNA collection, funded by the Medical Research Council grant G0000934 and the Wellcome Trust grant 068545/Z/02. Genotyping for the B58C-WTCCC subset was funded by the Wellcome Trust grant 076113/B/04/Z. The B58C-T1DGC genotyping utilized resources provided by the Type 1 Diabetes Genetics Consortium, a collaborative clinical study sponsored by the National Institute of Diabetes and Digestive and Kidney Diseases (NIDDK), National Institute of Allergy and Infectious Diseases (NIAID), National Human Genome Research Institute (NHGRI), National Institute of Child Health and Human Development (NICHD), and Juvenile Diabetes Research Foundation International (JDRF) and supported by U01 DK062418. B58C-T1DGC GWAS data were deposited by the Diabetes and Inflammation Laboratory, Cambridge Institute for Medical Research (CIMR), University of Cambridge, which is funded by Juvenile Diabetes Research Foundation International, the Wellcome Trust and the National Institute for Health Research Cambridge Biomedical Research Centre; the CIMR is in receipt of a Wellcome Trust Strategic Award (079895). The B58C-GABRIEL genotyping was supported by a contract from the European Commission Framework Programme 6 (018996) and grants from the French Ministry of Research. CHS: This CHS research was supported by NHLBI contracts HHSN268201200036C, HHSN268200800007C, N01HC55222, N01HC85079, N01HC85080, N01HC85081, N01HC85082, N01HC85083, N01HC85086, HHSN268200960009C; and NHLBI grants U01HL080295, R01HL087652, R01HL105756, R01HL103612, R01HL120393, and R01HL130114 with additional contribution from the National Institute of Neurological Disorders and Stroke (NINDS). Additional support was provided through R01AG023629 from the National Institute on Aging (NIA). A full list of principal CHS investigators and institutions can be found at CHS-. The provision of genotyping data was supported in part by the National Center for Advancing Translational Sciences, CTSI grant UL1TR000124, and the National Institute of Diabetes and Digestive and Kidney Disease Diabetes Research Center (DRC) grant DK063491 to the Southern California Diabetes Endocrinology Research Center. The content is solely the responsibility of the authors and does not necessarily represent the official views of the National Institutes of Health.Cilento study: The Cilento study was supported by the Italian Ministry of Education Universities and Research (Interomics Flagship Project, PON03PE_00060_7), FP6 (Vasoplus-037254), the Assessorato Ricerca Regione Campania, the Fondazione con il SUD (2011-PDR-13), and the Istituto Banco di Napoli - Fondazione to MC. We address special thanks to the populations of Cilento for their participation in the study.COLAUS: The CoLaus study was and is supported by research grants from GlaxoSmithKline (GSK), the Faculty of Biology and Medicine of Lausanne, and the Swiss National Science Foundation (grants 3200B0-105993, 3200B0- 118308, 33CSCO-122661, and 33CS30-139468). We thank all participants, involved physicians and study nurses to the CoLaus cohort.COROGENE_CTRL: This study has been funded by the Academy of Finland (grant numbers 139635, 129494, 118065, 129322, 250207), the Orion-Farmos Research Foundation, the Finnish Foundation for Cardiovascular Research, and the Sigrid Jusélius Foundation. We are grateful for the THL DNA laboratory for its skillful work to produce the DNA samples used in this study. We thank the Sanger Institute genotyping facilities for genotyping the samples.CROATIA Studies: The CROATIA-Vis, CROATIA-Korcula and CROATIA-Split studies in the Croatian islands of Vis and Korcula and mainland city of Split were supported by grants from the Medical Research Council (UK); the Ministry of Science, Education, and Sport of the Republic of Croatia (grant number 216-1080315-0302); the European Union framework program 6 European Special Populations Research Network project (contract LSHG-CT-2006-018947), the European Union framework program 7 project BBMRI-LPC (FP7 313010) and the Croatian Science Foundation (grant 8875). The CROATIA studies would like to acknowledge the invaluable contributions of the recruitment teams (including those from the Institute of Anthropological Research in Zagreb) in Vis, Korcula and Split, the administrative teams in Croatia and Edinburgh, and the people of Vis, Korcula and Split. SNP genotyping of the CROATIA-Vis samples was carried out by the Genetics Core Laboratory at the Wellcome Trust Clinical Research Facility, WGH, Edinburgh, Scotland. SNP genotyping for CROATIA-Korcula was performed by Helmholtz ZentrumMünchen, GmbH, Neuherberg, Germany. The SNP genotyping for the CROATIA-Split cohort was performed by AROS Applied Biotechnology, Aarhus, Denmark.ERF: The ERF study as a part of EUROSPAN (European Special Populations Research Network) was supported by European Commission FP6 STRP grant number 018947 (LSHG-CT-2006-01947) and also received funding from the European Community's Seventh Framework Programme (FP7/2007-2013)/grant agreement HEALTH-F4-2007-201413 by the European Commission under the programme "Quality of Life and Management of the Living Resources" of 5th Framework Programme (no. QLG2-CT-2002-01254). High-throughput analysis of the ERF data was supported by a joint grant from the Netherlands Organization for Scientific Research and the Russian Foundation for Basic Research (NWO-RFBR 047.017.043). Exome sequencing analysis in ERF was supported by the ZonMw grant (project 91111025). Najaf Amin is supported by the Netherlands Brain Foundation (project number F2013(1)-28). We are grateful to all study participants and their relatives, general practitioners and neurologists for their contributions and to P. Veraart for her help in genealogy, J. Vergeer for the supervision of the laboratory work and P. Snijders for his help in data collection.Fenland: JAL, CL, RAS and NJW acknowledge support from the Medical Research Council (MC_U106179471 and MC_UU_12015/1) The Fenland Study is funded by the Wellcome Trust and the Medical Research Council (MC_U106179471). We are grateful to all the volunteers for their time and help, and to the General Practitioners and practice staff for assistance with recruitment. We thank the Fenland Study Investigators, Fenland Study Co-ordination team and the Epidemiology Field, Data and Laboratory teams. We further acknowledge support from the Medical research council (MC_UU_12015/1). FHS: The National Heart, Lung and Blood Institute’s Framingham Heart Study is supported by contract N01-HC-25195 FINRISK_PREDICT_CVD: This study has been funded by the Academy of Finland (grant numbers 139635, 129494, 118065, 129322, 250207, 269517), the Orion-Farmos Research Foundation, the Finnish Foundation for Cardiovascular Research, and the Sigrid Jusélius Foundation. We are grateful for the THL DNA laboratory for its skillful work to produce the DNA samples used in this study. We thank the Sanger Institute genotyping facilities for genotyping the samples.FUSION: Support for FUSION was provided by NIH grants R01-DK062370 (to M.B.) and intramural project number ZIA-HG000024 (to F.S.C.). Genome-wide genotyping was conducted by the Johns Hopkins University Genetic Resources Core Facility SNP Center at the Center for Inherited Disease Research (CIDR), with support from CIDR NIH contract no. N01-HG-65403.GAPP study: The GAPP study was supported by the Liechtenstein Government,?the Swiss National Science?Foundation,?the Swiss Heart Foundation, the Swiss Society of Hypertension, the University of Basel, the University Hospital Basel, the?Hanela?Foundation, Schiller AG and Novartis.GS:SFHS: Generation Scotland received core support from the Chief Scientist Office of the Scottish Government Health Directorates [CZD/16/6] and the Scottish Funding Council [HR03006]. Genotyping of the GS:SFHS samples was carried out by the Genetics Core Laboratory at the Wellcome Trust Clinical Research Facility, Edinburgh, Scotland and was funded by the Medical Research Council UK and the Wellcome Trust (Wellcome Trust Strategic Award “STratifying Resilience and Depression Longitudinally” (STRADL) Reference 104036/Z/14/Z). Ethics approval for the study was given by the NHS Tayside committee on research ethics (reference 05/S1401/89). We are grateful to all the families who took part, the general practitioners and the Scottish School of Primary Care for their help in recruiting them, and the whole Generation Scotland team, which includes interviewers, computer and laboratory technicians, clerical workers, research scientists, volunteers, managers, receptionists, healthcare assistants and nurses.GoDARTS: GoDARTS was funded by The Wellcome Trust (072960/Z/03/Z, 084726/Z/08/Z, 084727/Z/08/Z, 085475/Z/08/Z, 085475/B/08/Z) and as part of the EU IMI-SUMMIT program. We acknowledge the support of the Health Informatics Centre, University of Dundee for managing and supplying the anonymised data and NHS Tayside, the original data owner. We are grateful to all the participants who took part in the Go-DARTS study, to the general practitioners, to the Scottish School of Primary Care for their help in recruiting the participants, and to the whole team, which includes interviewers, computer and laboratory technicians, clerical workers, research scientists, volunteers, managers, receptionists, and nurses. GRAPHIC: The GRAPHIC Study was funded by the British Heart Foundation (BHF/RG/2000004). CPN and NJS are supported by the British Heart Foundation and NJS is a NIHR Senior Investigator This work falls under the portfolio of research supported by the NIHR Leicester Cardiovascular Biomedical Research Unit.H2000: The Health 2000 Study was funded by the National Institute for Health and Welfare (THL), the Finnish Centre for Pensions (ETK), the Social Insurance Institution of Finland (KELA), the Local Government Pensions Institution (KEVA) and other organizations listed on the website of the survey ( ). We are grateful for the THL DNA laboratory for its skillful work to produce the DNA samples used in this study. We thank the Sanger Institute genotyping facilities for genotyping the GenMets subcohort.HABC: The Health ABC Study was supported by NIA contracts N01AG62101, N01AG62103, and N01AG62106 and, in part, by the NIA Intramural Research Program. The genome-wide association study was funded by NIA grant 1R01AG032098-01A1 to Wake Forest University Health Sciences and genotyping services were provided by the Center for Inherited Disease Research (CIDR). CIDR is fully funded through a federal contract from the National Institutes of Health to The Johns Hopkins University, contract number HHSN268200782096C. This study utilized the high-performance computational capabilities of the Biowulf Linux cluster at the National Institutes of Health, Bethesda, Md. (). HTO: The study was funded by the Wellcome Trust, Medical Research Council and British Heart Foundation We thank all the families who participated in the studyINGI-VB: The INGI‐Val Borbera population is a collection of 1,664 genotyped samples collected in the Val Borbera Valley, a geographically isolated valley located within the Appennine Mountains in Northwest Italy. The valley is inhabited by about 3,000 descendants from the original population, living in 7 villages along the valley and in the mountains. Participants were healthy people 18-102 years of age that had at least one grandfather living in the valley. The study plan and the informed consent form were reviewed and approved by the institutional review boards of San Raffaele Hospital in Milan. The research was supported by funds from Compagnia di San Paolo, Torino, Italy; Fondazione Cariplo, Italy and Ministry of Health, Ricerca Finalizzata 2008 and CCM 2010, PRIN 2009 and Telethon, Italy to DT. The funders had no role in study design, data collection and analysis, decision to publish, or preparation of the manuscript. We thank the inhabitants of the VB that made this study possible, the local administrations, the MD of the San Raffaele Hospital and Prof Clara Camaschella for clinical data collection. We also thank Fiammetta Vigano? for technical help, Corrado Masciullo and Massimiliano Cocca for building and maintaining the analysis platform.INGI-CARL: Italian Ministry of Health RF2010 to Paolo Gasparini, RC2008 to Paolo Gasparini INGI-FVG: Italian Ministry of Health RF2010 to Paolo Gasparini, RC2008 to Paolo Gasparini JUPITER: Genetic analysis in the JUPITER trial was funded by a grant from AstraZeneca (DIC and PMR, Co-Pis). KORA S3: KORA S3 500K blood pressure project was supported by Estonian Research Council, grant IUT34-12 (for Maris Laan). The KORA Augsburg studies have been financed by the Helmholtz Zentrum Mu nchen, German Research Center for Environmental Health, Neuherberg, Germany and supported by grants from the German Federal Ministry of Education and Research (BMBF). The KORA study group consists of H-E. Wichmann (speaker), A. Peters, C. Meisinger, T. Illig, R. Holle, J. John and co-workers, who are responsible for the design and conduct of the KORA studies. Part of this work was financed by the German National Genome Research Network (NGFN-2 and NGFNPlus:01GS0823) and supported within the Munich Center of Health Sciences (MC Health) as part of LMUinnovativ. LBC1921: Phenotype collection in the Lothian Birth Cohort 1921 was supported by the UK’s Biotechnology and Biological Sciences Research Council (BBSRC), The Royal Society, and The Chief Scientist Office of the Scottish Government. Genotyping was funded by the BBSRC. The work was undertaken by The University of Edinburgh Centre for Cognitive Ageing and Cognitive Epidemiology, part of the cross council Lifelong Health and Wellbeing Initiative (MR/K026992/1). Funding from the BBSRC and Medical Research Council (MRC) is gratefully acknowledged. We thank the Lothian Birth Cohort 1921 participants and team members who contributed to these studies.LBC1936: Phenotype collection in the Lothian Birth Cohort 1936 was supported by Age UK (The Disconnected Mind project).? Genotyping was funded by the BBSRC. The work was undertaken by The University of Edinburgh Centre for Cognitive Ageing and Cognitive Epidemiology, part of the cross council Lifelong Health and Wellbeing Initiative (MR/K026992/1). Funding from the BBSRC and Medical Research Council (MRC) is gratefully acknowledged. We thank the Lothian Birth Cohort 1936 participants and team members who contributed to these studies.Lifelines Cohort Study: The LifeLines Cohort Study, and generation and management of GWAS genotype data for the LifeLines Cohort Study is supported by the Netherlands Organization of Scientific Research NWO (grant 175.010.2007.006), the Economic Structure Enhancing Fund (FES) of the Dutch government, the Ministry of Economic Affairs, the Ministry of Education, Culture and Science, the Ministry for Health, Welfare and Sports, the Northern Netherlands Collaboration of Provinces (SNN), the Province of Groningen, University Medical Center Groningen, the University of Groningen, Dutch Kidney Foundation and Dutch Diabetes Research Foundation. The authors wish to acknowledge the services of the Lifelines Cohort Study, the contributing research centers delivering data to Lifelines, and all the study participants.LOLIPOP: The LOLIPOP study is funded by the British Heart Foundation (SP/04/002), the Medical Research Council (G0601966, G0700931), the Wellcome Trust (084723/Z/08/Z), the NIHR (RP-PG-0407-10371), European Union FP7 (EpiMigrant, 279143) and Action on Hearing Loss (G51). The LOLIPOP study is supported by the National Institute for Health Research (NIHR) Comprehensive Biomedical Research Centre Imperial College Healthcare NHS Trust. The work was carried out in part at the NIHR/Wellcome Trust Imperial Clinical Research Facility. We thank the participants and research staff who made the study possible.MESA: This research was supported by the Multi-Ethnic Study of Atherosclerosis (MESA) contracts N01-HC-95159, N01-HC-95160, N01-HC-95161, N01-HC-95162, N01-HC-95163, N01-HC-95164, N01-HC-95165, N01-HC-95166, N01-HC-95167, N01-HC-95168, N01-HC-95169 and by grants UL1-TR-000040 and UL1-RR-025005 from NCRR . Funding for MESA SHARe genotyping was provided by NHLBI Contract N02-HL-6-4278. The provision of genotyping data was supported in part by the National Center for Advancing Translational Sciences, CTSI grant UL1TR000124, and the National Institute of Diabetes and Digestive and Kidney Disease Diabetes Research Center (DRC) grant DK063491 to the Southern California Diabetes Endocrinology Research Center. MICROS: The MICROS study was supported by the Ministry of Health and Department of Innovation, Research and University of the Autonomous Province of Bolzano, the South Tyrolean Sparkasse Foundation, and the European Union framework program 6 EUROSPAN project (contract no. LSHG-CT-2006-018947) For the MICROS study, we thank the primary care practitioners Raffaela Stocker, Stefan Waldner, Toni Pizzecco, Josef Plangger, Ugo Marcadent, and the personnel of the Hospital of Silandro (Department of Laboratory Medicine) for their participation and collaboration in the research project.NEO: The NEO study is supported by the participating Departments, the Division and the Board of Directors of the Leiden University Medical Center, and by the Leiden University, Research Profile Area Vascular and Regenerative Medicine. Dennis Mook-Kanamori is supported by Dutch Science Organization (ZonMW-VENI Grant 916.14.023). The authors of the NEO study thank all individuals who participated in the Netherlands Epidemiology in Obesity study, all participating general practitioners for inviting eligible participants and all research nurses for collection of the data. We thank the NEO study group, Pat van Beelen, Petra Noordijk and Ingeborg de Jonge for the coordination, lab and data management of the NEO study. The genotyping in the NEO study was supported by the Centre National de Génotypage (Paris, France), headed by Jean-Francois Deleuze. NESDA: Funding was obtained from the Netherlands Organization for Scientific Research (Geestkracht program grant 10-000-1002); the Center for Medical Systems Biology (CSMB, NOW Genomics), Biobanking and Biomolecular Resources Research Infrastructure (BBMRI-NL), VU University’s Institutes for Health and Care Research (EMGO+) and Neuroscience Campus Amsterdam, University Medical Center Groningen, Leiden University Medical Center, National Institutes of Health (NIH, R01D0042157-01A, MH081802, Grand Opportunity grants 1RC2 MH089951 and 1RC2 MH089995). Part of the genotyping and analyses were funded by the Genetic Association Information Network (GAIN) of the Foundation for the National Institutes of Health. Computing was supported by BiG Grid, the Dutch e-Science Grid, which is financially supported by NWO.NSPHS: The Northern Swedish Population Health Study (NSPHS) was funded by the Swedish Medical Research Council (Project Number K2007-66X-20270-01-3, 2011-5252, 2012-2884 and 2011-2354), the Foundation for Strategic Research (SSF). NSPHS as part of EUROSPAN (European Special Populations Research Network) was also supported by the European Commission FP6 STRP grant number 01947 (LSHG-CT-2006-01947). This work has also been supported by the Swedish Society for Medical Research (SSMF), and the Swedish Medical Research Council (#2015-03327) We are grateful for the contribution of district nurse Svea Hennix for data collection and Inger Jonasson for logistics and coordination of the health survey. We also thank all the participants from the community for their interest and willingness to contribute to this study. NTR: Funding was obtained from the Netherlands Organization for Scientific Research (NWO) and The Netherlands Organisation for Health Research and Development (ZonMW) grants 904-61-090, 985-10-002, 904-61-193,480-04-004, 400-05-717, Addiction-31160008, Middelgroot-911-09-032, Spinozapremie 56-464-14192, Biobanking and Biomolecular Resources Research Infrastructure (BBMRI –NL, 184.021.007); the Netherlands Heart Foundation grants 86.083 and 88.042 and 90.313; the VU Institute for Health and Care Research (EMGO+ ); the European Community's Seventh Framework Program (FP7/2007-2013), ENGAGE (HEALTH-F4-2007-201413); the European Research Council (ERC Advanced, 230374), the Rutgers University Cell and DNA Repository (NIMH U24 MH068457-06), the Avera Institute, Sioux Falls, South Dakota (USA) and the National Institutes of Health (NIH, R01D0042157-01A, MH081802; Grand Opportunity grant 1RC2 MH089951). Part of the genotyping and analyses were funded by the Genetic Association Information Network (GAIN) of the Foundation for the National Institutes of Health. Computing was supported by BiG Grid, the Dutch e-Science Grid, which is financially supported by NWO. "ORCADES: ORCADES was supported by the Chief Scientist Office of the Scottish Government, the Royal Society, the MRC Human Genetics Unit, Arthritis Research UK and the European Union framework program 6 EUROSPAN project (contract no. LSHG-CT-2006-018947). DNA extractions were performed at the Wellcome Trust Clinical Research Facility in Edinburgh. We would like to acknowledge the invaluable contributions of Lorraine Anderson and the research nurses in Orkney, the administrative team in Edinburgh and the people of Orkney.PIVUS: This project was supported by Knut and Alice Wallenberg Foundation (Wallenberg Academy Fellow), European Research Council (ERC Starting Grant), Swedish Diabetes Foundation (grant no. 2013-024), Swedish Research Council (grant no. 2012-1397), and Swedish Heart-Lung Foundation (20120197). The computations were performed on resources provided by SNIC through Uppsala Multidisciplinary Center for Advanced Computational Science (UPPMAX) under Project b2011036. Genetic data analysis was funded by the Wellcome Trust under awards WT098017 and WT090532. We thank the SNP&SEQ Technology Platform in Uppsala (genotyping.se) for excellent genotyping. PROCARDIS: PROCARDIS was supported by the European Community Sixth Framework Program (LSHM-CT- 2007-037273), AstraZeneca, the British Heart Foundation, the Swedish Research Council, the Knut and Alice Wallenberg Foundation, the Swedish Heart-Lung Foundation, the Torsten and Ragnar S?derberg Foundation, the Strategic Cardiovascular Program of Karolinska Institutet and Stockholm County Council, the Foundation for Strategic Research and the Stockholm County Council (560283). M.F and H.W acknowledge the support of the Wellcome Trust core award (090532/Z/09/Z) and M.F, H.W, the BHF Centre of Research Excellence (RE/13/1/30181). A.G, H.W acknowledge European Union Seventh Framework Programme FP7/2007-2013 under grant agreement no. HEALTH-F2-2013-601456 (CVGenes@Target) & and A.G, the Wellcome Trust Institutional strategic support fund. PROCARDIS was supported by the European Community Sixth Framework Program (LSHM-CT- 2007-037273), AstraZeneca, the British Heart Foundation, the Swedish Research Council, the Knut and Alice Wallenberg Foundation, the Swedish Heart-Lung Foundation, the Torsten and Ragnar S?derberg Foundation, the Strategic Cardiovascular Program of Karolinska Institutet and Stockholm County Council, the Foundation for Strategic Research and the Stockholm County Council (560283). M.F and H.W acknowledge the support of the Wellcome Trust core award (090532/Z/09/Z) and M.F, H.W, the BHF Centre of Research Excellence (RE/13/1/30181). A.G, H.W acknowledge European Union Seventh Framework Programme FP7/2007-2013 under grant agreement no. HEALTH-F2-2013-601456 (CVGenes@Target) & and A.G, the Wellcome Trust Institutional strategic support fund. PROSPER: The PROSPER study was supported by an investigator initiated grant obtained from Bristol-Myers Squibb. Prof. Dr. J. W. Jukema is an Established Clinical Investigator of the Netherlands Heart Foundation (grant 2001 D 032). Support for genotyping was provided by the seventh framework program of the European commission (grant 223004) and by the Netherlands Genomics Initiative (Netherlands Consortium for Healthy Aging grant 050-060-810). RS: The generation and management of GWAS genotype data for the Rotterdam Study (RS I, RS II, RS III) was executed by the Human Genotyping Facility of the Genetic Laboratory of the Department of Internal Medicine, Erasmus MC, Rotterdam, The Netherlands. The GWAS datasets are supported by the Netherlands Organisation of Scientific Research NWO Investments (nr. 175.010.2005.011, 911-03-012), the Genetic Laboratory of the Department of Internal Medicine, Erasmus MC, the Research Institute for Diseases in the Elderly (014-93-015; RIDE2), the Netherlands Genomics Initiative (NGI)/Netherlands Organisation for Scientific Research (NWO) Netherlands Consortium for Healthy Aging (NCHA), project nr. 050-060-810. The Rotterdam Study is funded by Erasmus Medical Center and Erasmus University, Rotterdam, Netherlands Organization for the Health Research and Development (ZonMw), the Research Institute for Diseases in the Elderly (RIDE), the Ministry of Education, Culture and Science, the Ministry for Health, Welfare and Sports, the European Commission (DG XII), and the Municipality of Rotterdam. We thank Pascal Arp, Mila Jhamai, Marijn Verkerk, Lizbeth Herrera and Marjolein Peters, MSc, and Carolina Medina-Gomez, MSc, for their help in creating the GWAS database, and Karol Estrada, PhD, Yurii Aulchenko, PhD, and Carolina Medina-Gomez, MSc, for the creation and analysis of imputed data.The authors are grateful to the study participants, the staff from the Rotterdam Study and the participating general practitioners and pharmacists. SHIP: SHIP is part of the Community Medicine Research net of the University of Greifswald, Germany, which is funded by the Federal Ministry of Education and Research (grants no. 01ZZ9603, 01ZZ0103, and 01ZZ0403), the Ministry of Cultural Affairs as well as the Social Ministry of the Federal State of Mecklenburg-West Pomerania, and the network ‘Greifswald Approach to Individualized Medicine (GANI_MED)’ funded by the Federal Ministry of Education and Research (grant 03IS2061A). Genome-wide data have been supported by the Federal Ministry of Education and Research (grant no. 03ZIK012) and a joint grant from Siemens Healthcare, Erlangen, Germany and the Federal State of Mecklenburg- West Pomerania. The University of Greifswald is a member of the Caché Campus program of the InterSystems GmbH. Three City- Dijon: The 3-City Study is conducted under a partnership agreement among the Institut National de la Santé et de la Recherche Médicale (INSERM), the University of Bordeaux, and Sanofi-Aventis. The Fondation pour la Recherche Médicale funded the preparation and initiation of the study. The 3C Study is also supported by the Caisse Nationale Maladie des Travailleurs Salariés, Direction Générale de la Santé, Mutuelle Générale de l’Education Nationale (MGEN), Institut de la Longévité, Conseils Régionaux of Aquitaine and Bourgogne, Fondation de France, and Ministry of Research–INSERM Programme “Cohortes et collections de données biologiques.” This work was supported by the National Foundation for Alzheimer’s Disease and Related Disorders, the Institut Pasteur de Lille, the Centre National de Génotypage and the LABEX (Laboratory of Excellence program investment for the future) DISTALZ - Development of Innovative Strategies for a Transdisciplinary approach to ALZheimer’s disease. Ganesh Chauhan, Christophe Tzourio and Stéphanie Debette are supported by a grant from the Fondation Leducq. We thank Philippe Amouyel and the UMR1167 Inserm Univ Lille Institut Pasteur de Lille for providing the 3C Dijon cohort SNP replication data funded by a grant from the French National Foundation on Alzheimer’s disease and related disorders.UKHLS: This work was funded through generous grants from the Economic & Social Research Council (ES/H029745/1) and the Wellcome Trust (WT098051). TRAILS: This research is part of the TRacking Adolescents' Individual Lives Survey (TRAILS). Participating centers of TRAILS include the University Medical Center and University of Groningen, the Erasmus University Medical Center Rotterdam, the University of Utrecht, the Radboud Medical Center Nijmegen, and the Parnassia Bavo group, all in the Netherlands. TRAILS has been financially supported by various grants from the Netherlands Organization for Scientific Research NWO (Medical Research Council program grant GB-MW 940-38-011; ZonMW Brainpower grant 100-001-004; ZonMw Risk Behavior and Dependence grants 60-60600-97-118; ZonMw Culture and Health grant 261-98-710; Social Sciences Council medium-sized investment grants GB-MaGW 480-01-006 and GB-MaGW 480-07-001; Social Sciences Council project grants GB-MaGW 452-04-314 and GB-MaGW 452-06-004; NWO large-sized investment grant 175.010.2003.005; NWO Longitudinal Survey and Panel Funding 481-08-013 and 481-11-001), the Dutch Ministry of Justice (WODC), the European Science Foundation (EuroSTRESS project FP-006), Biobanking and Biomolecular Resources Research Infrastructure BBMRI-NL (CP 32), and the participating universities. Statistical analyses were carried out on the Genetic Cluster Computer () hosted by SURFsara and financially supported by the Netherlands Scientific Organization (NWO 480-05-003 PI: Posthuma) along with a supplement from the Dutch Brain Foundation and the VU University Amsterdam.TwinGene: This project was supported by grants from the Ministry for Higher Education, the Swedish Research Council (M-2005-1112 and 2009-2298), GenomEUtwin (EU/QLRT-2001-01254; QLG2-CT-2002-01254), NIH grant DK U01-066134, Knut and Alice Wallenberg Foundation (Wallenberg Academy Fellow), European Research Council (ERC Starting Grant), Swedish Diabetes Foundation (grant no. 2013-024), Swedish Research Council (grant no. 2012-1397), and Swedish Heart-Lung Foundation (20120197). We thank the SNP&SEQ Technology Platform in Uppsala (genotyping.se) for excellent genotyping. The computations were performed on resources provided by SNIC through Uppsala Multidisciplinary Center for Advanced Computational Science (UPPMAX) under Project b2011036.TwinsUK: The study was funded by the Wellcome Trust; European Community’s Seventh Framework Programme (FP7/2007-2013). The study also receives support from the National Institute for Health Research (NIHR) BioResource Clinical Research Facility and Biomedical Research Centre based at Guy's and St Thomas' NHS Foundation Trust and King's College London (guysbrc-2012-1). We thank the staff from the Genotyping Facilities at the Wellcome Trust Sanger Institute for sample preparation, quality control, and genotyping; Le Centre National de Génotypage, France, for genotyping; Duke University, NC, USA, for genotyping; and the Finnish Institute of Molecular Medicine, Finnish Genome Center, University of Helsinki. Genotyping was also done by CIDR as part of an NEI/NIH project grantUK Biobank_Cardiometabolic Consortium: This research has been conducted using the UK Biobank Resource under application number 236. H.R.W., C.P.C and M.R.B. were funded by the National Institutes for Health Research (NIHR) as part of the portfolio of translational research of the NIHR Biomedical Research Unit at Barts MR was funded by the National Institute for Health Research (NIHR) Biomedical Research Unit in Cardiovascular Disease at Barts. MR is recipient from China Scholarship Council (No. 2011632047). B.M. holds an MRC?eMedLab?Medical Bioinformatics Career Development Fellowship, funded from award MR/L016311/1. PE was funded by the National Institutes for Health Research (NIHR) Imperial College Health Care NHS Trust and Imperial College London Biomedical Research Centre, the UK Medical Research Council and Public Health England as Director of the MRC-PHE Centre for Environment and Health, and the NIHR Health Protection Research Unit on the Health Effects of Environmental Hazards. Some of this work used computing resources provided by the Medical Research Council-funded UK MEDical Bioinformatics partnership programme (UK MED-BIO) (MR/L01632X/1). ULSAM: This project was supported by Knut and Alice Wallenberg Foundation (Wallenberg Academy Fellow), European Research Council (ERC Starting Grant), Swedish Diabetes Foundation (grant no. 2013-024), Swedish Research Council (grant no. 2012-1397), and Swedish Heart-Lung Foundation (20120197). The computations were performed on resources provided by SNIC through Uppsala Multidisciplinary Center for Advanced Computational Science (UPPMAX) under Project b2011036. Genotyping was funded by the Wellcome Trust under award WT064890. Analysis of genetic data was funded by the Wellcome Trust under awards WT098017 and WT090532. Andrew P. Morris is a Wellcome Trust Senior Research Fellow in Basic Biomedical Science (WT098017). We thank the SNP&SEQ Technology Platform in Uppsala (genotyping.se) for excellent genotyping. WGHS: The WGHS is supported by the National Heart, Lung, and Blood Institute (HL043851, HL080467, HL09935) and the National Cancer Institute (CA047988 and UM1CA182913) with collaborative scientific support and funding for genotyping provided by Amgen. YFS: The Young Finns Study has been financially supported by the Academy of Finland: grants 286284, 134309 (Eye), 126925, 121584, 124282, 129378 (Salve), 117787 (Gendi), and 41071 (Skidi); the Social Insurance Institution of Finland; Kuopio, Tampere and Turku University Hospital Medical Funds (grant X51001); Juho Vainio Foundation; Paavo Nurmi Foundation; Finnish Foundation for Cardiovascular Research ; Finnish Cultural Foundation; Tampere Tuberculosis Foundation; Emil Aaltonen Foundation; Yrj? Jahnsson Foundation; Signe and Ane Gyllenberg Foundation; and Diabetes Research Foundation of Finnish Diabetes Association. The expert technical assistance in the statistical analyses by Irina Lisinen is gratefully acknowledged. ................
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